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N-cyclohexyl-4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
1-[4-(furan-2-ylmethyl)-6-hydroxy-1,4-diazepan-1-yl]-2-(1H-imidazol-4-yl)ethan-1-one
2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxamide
7-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[1-phenyl-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]benzene-1,3-diol
1-(cyclopropylmethyl)-4-[(2,4-diethoxy-3-methylphenyl)methyl]piperazine
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}propanamide
5-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-(1,2-oxazol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
3-[5-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
3-methyl-5-(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,2-oxazole
ethyl 2-{1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidin-2-yl}acetate
5-{[methyl(oxan-4-ylmethyl)amino]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
2-(3,4-dimethoxyphenyl)-1-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-4-yl)-1H-1,3-benzodiazole
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}propanamide
N-[(2S)-1-{2-tert-butyl-4-oxo-1,3,8-triazaspiro[4.5]dec-1-en-8-yl}-4-methyl-1-oxopentan-2-yl]acetamide
6-ethyl-2-(morpholin-4-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}pyrimidin-4-amine
2-cyclopropyl-4-methyl-5-(3-methyl-3-phenylpiperidine-1-carbonyl)pyrimidine
N4-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[4-(trifluoromethyl)phenyl]methyl}acetamide
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-chlorophenyl)urea
2-(benzyloxy)-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}ethan-1-one
5-chloro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-7-methoxy-1-benzofuran-2-carboxamide
(3S,4S)-1-[(4-methyl-1H-imidazol-2-yl)methyl]-4-(piperidin-1-yl)pyrrolidin-3-ol
2-{2-[(3S)-3-acetamidopyrrolidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
5-(methoxymethyl)-N-({7-[(6-methylpyridin-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)furan-2-carboxamide
1-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-2-(pyridin-3-yloxy)ethan-1-one
2-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]pyrimidin-4-amine
N1,N1-dimethyl-N3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-1,3-dicarboxamide
2-amino-N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
[(4,6-dimethylpyridin-2-yl)methyl](methyl)({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
3-(5-{[2-(difluoromethoxy)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl)pyridine
1-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-N-cyclopropylpiperazine-2-carboxamide
(3S,4R)-4-(2-methoxyphenyl)-1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)pyrrolidine-3-carboxylic acid
(3R,4R)-3-cyclopropyl-1-(2-methoxyquinoline-4-carbonyl)-4-methylpyrrolidin-3-ol
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
9-[(4-acetylphenyl)methyl]-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl[1-(1,2-oxazol-3-yl)ethyl][(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
N-[(2,6-difluorophenyl)methyl]-2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]acetamide
1,4-dimethyl-9-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-1,4,9-triazaspiro[5.5]undecane
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-5,6-dimethylpyrimidin-4-amine
5-ethyl-2-methyl-4-{4-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}pyrimidine
2-ethyl-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1-(propan-2-yl)piperazine
N-{1-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-2-phenylethyl}-N,2-dimethylfuran-3-carboxamide
N-[(cyclopropylcarbamoyl)methyl]-2-(dimethylamino)-2-(3-methylphenyl)acetamide
3-({3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}methoxy)pyridine
1-[(3-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}-4-methoxyphenyl)methyl]piperidin-4-ol
3-{[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]sulfamoyl}-N-pentylbenzamide
N-ethyl-8-[(4-methylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
2-(9H-carbazol-3-yl)-1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one