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N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(quinoxalin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-1λ6-thiomorpholine-1,1-dione
N-[2-(diethylamino)ethyl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
7-fluoro-3-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-1-[2-(piperidin-1-yl)ethyl]-1,2-dihydroquinolin-2-one
2,4-dimethyl-N-(4-{4-[(oxan-4-ylmethyl)amino]piperidin-1-yl}phenyl)benzamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[2-(oxan-2-yl)ethyl]-1,2-oxazole-3-carboxamide
(4aS,7aR)-1-[(5-propylfuran-2-yl)methyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-{3-[1-(dimethylamino)ethyl]phenyl}-2,3-dihydro-1H-inden-1-one
(3R,5S)-N-(2-methylpropyl)-5-(morpholin-4-ylmethyl)piperidine-3-carboxamide
3-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-(4-methylpiperidin-1-yl)propan-1-one
6-[(3R,5S)-5-(morpholine-4-carbonyl)piperidine-3-carbonyl]-5,6,7,8-tetrahydro-1,6-naphthyridine
2-[3-(furan-2-yl)-5-(1-methyl-3-propyl-1H-pyrazol-5-yl)-1H-1,2,4-triazol-1-yl]acetic acid
1-(6-oxopiperazine-2-carbonyl)-4-phenylpiperidine-4-carbonitrile
4-[1-(4-chlorophenyl)cyclobutanecarbonyl]-9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2S,4S)-4-[2-amino-6-(propan-2-yl)pyrimidine-4-amido]-1-methylpyrrolidine-2-carboxylic acid
1-(1-{6-[(furan-3-ylmethyl)(methyl)amino]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
3-(6-chloropyridin-3-yl)-1-(oxolan-2-ylmethyl)-1-(2-phenoxyethyl)urea
4-benzyl-3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-hydroxyethyl)-N-(1-phenylethyl)-5-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propanamide
(2-methoxyethyl)({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})(propan-2-yl)amine
1-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-3-(3-methyl-1-phenyl-1H-pyrazol-5-yl)urea
N-(2,1,3-benzoxadiazol-5-ylmethyl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)pyridine
N-benzyl-N-(1,3-thiazol-2-ylmethyl)cyclohex-3-ene-1-carboxamide
(3R,4S)-1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-3,4-dimethylpiperidin-4-ol
2-methyl-6-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
1-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-6-[(4-phenylpiperidin-1-yl)methyl]-1,2-dihydropyridine-3-carboxamide
N-{[(2S,4S)-1-[5-(ethylsulfanyl)thiophene-2-carbonyl]-4-fluoropyrrolidin-2-yl]methyl}cyclobutanecarboxamide
methyl[(3-methyl-1,2-oxazol-5-yl)methyl]({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)amine
5-benzyl-5-(1-{2-[3-(trifluoromethyl)phenyl]acetyl}piperidin-4-yl)imidazolidine-2,4-dione
(3S,9R)-11-[4-(trifluoromethyl)benzoyl]-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
3-chloro-4-fluoro-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-benzothiophene-2-carboxamide
1-(1-ethyl-1H-pyrazole-5-carbonyl)-4-(2-methoxyphenoxy)piperidine
N-benzyl-1-[(2-chlorophenyl)methyl]-N-(2-hydroxyethyl)-1H-1,2,3-triazole-4-carboxamide
(3aS,6aS)-2-cyclopentyl-5-(pyrazin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{2-[(7-fluoro-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-6-methylpyrimidin-2-amine
2-(5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)pyridine
2-amino-6-(3,5-difluorophenyl)-4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-{3-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[({5-[1-(2,2,2-trifluoroethyl)-1H-pyrazol-3-yl]furan-2-yl}methyl)amino]propan-2-ol
1-{[5-(methoxymethyl)furan-2-yl]methyl}-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)pyrrolidin-3-yl]methanol
9-[2-(2,5-dimethylphenyl)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
ethyl 1-(4-methylphenyl)-5-(pyrrolidin-1-ylmethyl)-1H-pyrazole-4-carboxylate
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide