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N-[2-(3-ethylphenoxy)ethyl]-N-methylspiro[2.2]pentane-1-carboxamide
2-(2,3-dimethylphenoxy)-N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]acetamide
3-(4-methyl-1,3-thiazol-5-yl)-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}propanamide
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]acetamide
dimethyl(3-{2-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
1-{4-[(dimethylamino)methyl]-2-methoxyphenoxy}-3-(4-ethylpiperazin-1-yl)propan-2-ol
N-[3-(2-chlorophenoxy)propyl]-N-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
6-methoxy-N-{[3-(morpholin-4-ylmethyl)phenyl]methyl}-1,3-benzothiazol-2-amine
5-{4-[(ethylcarbamoyl)amino]phenyl}-N,N-dimethylthiophene-2-carboxamide
(2S,4R)-4-amino-1-[(5-cyclohexylthiophen-2-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(3-methyl-1,2-thiazol-5-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
4-{4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-1-yl}quinazoline
ethyl 1-[1-(methylsulfanyl)propan-2-yl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-{2-[1-(3,4-dimethoxybenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
4-[4-(dimethylamino)phenyl]-1-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-{5-[1-(morpholin-4-yl)cyclohexanecarbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
(4aS,8aR)-6-(1H-1,3-benzodiazol-2-ylmethyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
(3aR,6aR)-2-acetyl-N-[2-(pyridin-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
4-fluoro-3-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]benzene-1-sulfonamide
1-(1-benzylpiperidin-4-yl)-N-butyl-N-methylpiperidine-3-carboxamide
1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylethan-1-one
4-phenyl-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}-1,2,3,6-tetrahydropyridine
7-(5-chloropyridine-2-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-[4-(2-methylpyrimidine-5-carbonyl)piperazin-1-yl]-6-phenyl-2,3-dihydropyridazin-3-one
[(2S)-1-{5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-2-yl]methanol
N-methyl-N-[2-({2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)ethyl]methanesulfonamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(pyridin-3-yloxy)ethyl]piperidine-4-carboxamide
8-(5-fluoro-2-methylbenzenesulfonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
methyl (2S,4S)-1-[(2,5-dimethylphenyl)methyl]-4-acetamidopyrrolidine-2-carboxylate
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperazine
1-[4-(furan-2-yl)butan-2-yl]-4-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazole
8-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-benzyl-8-(5-propyl-1,2-oxazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
7,7-dimethyl-2-[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(3S,4R)-1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
dimethyl(2-{4-[(2-phenyl-1,3-thiazol-5-yl)methyl]morpholin-2-yl}ethyl)amine
5-{1-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-imidazol-2-yl}-2,1,3-benzoxadiazole
4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]pyrimidin-2-amine
2-(4-methyl-1,4-diazepan-1-yl)-N-[(4-methylphenyl)(pyridin-4-yl)methyl]acetamide
2-methyl-4-[3-(1,2,3,6-tetrahydropyridine-1-carbonyl)phenyl]but-3-yn-2-ol
2-(3-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
3-fluoro-5-[3-(3-methylbutyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl]benzonitrile
4-(2-methyl-1H-imidazol-1-yl)-1-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperidine-4-carboxylic acid
4-[3-(2-chloro-6-methoxyphenyl)phenyl]-4H-1,2,4-triazole
6-methoxy-2-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,2,3,4-tetrahydroisoquinoline
1-{[1-butyl-2-(cyclohexanesulfonyl)-1H-imidazol-5-yl]methyl}-2-(2-methoxyethyl)piperidine
N-(1-cyclohexyl-1H-pyrazol-5-yl)-3-cyclopropylpropanamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-(furan-2-yl)-2-oxoacetamide
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-N-[3-(morpholin-4-yl)propyl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide