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ethyl 1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
3-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-3-methyl-1-[4-(oxan-2-ylmethoxy)phenyl]urea
(2R)-2-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-3-phenylpropan-1-ol
1-[3-(benzylsulfanyl)propyl]-3-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
methyl[(3-methylpyridin-4-yl)methyl]{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}amine
1-{1-[1-(2-chloro-4-fluorobenzoyl)piperidin-4-yl]ethyl}-4-methylpiperazine
5-[6-amino-5-cyano-4-(4-hydroxy-2-methoxyphenyl)pyridin-2-yl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyridin-2-yl)ethyl]amine
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-methyl-3-(propan-2-yl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
3-[(4aR,7aS)-4-[(3-methylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-{[7-fluoro-5-(quinolin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)acetamide
2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-4-(pyridin-3-yl)pyrimidine
1-(prop-2-en-1-yl)-N-[3-(propan-2-yloxy)propyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-methyl-2-{[3-(5-methylfuran-2-yl)-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl](methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
1-(4-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
N1,N1-dimethyl-N3-[(6-methylquinolin-5-yl)methyl]piperidine-1,3-dicarboxamide
N-[(7-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-2-phenylacetamide
2-(butylsulfanyl)-6-(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)pyrimidin-4-amine
N-(cyclopent-3-en-1-yl)-2-(4-{2-[(cyclopropylmethyl)sulfanyl]acetyl}morpholin-3-yl)acetamide
1-(4-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
3-{1-[(2-cyanophenyl)methyl]piperidin-4-yl}-N-[(4-fluorophenyl)methyl]propanamide
5-{[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]carbamoyl}-2,1,3-benzoxadiazol-1-ium-1-olate
ethyl 4-{[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate
4-hydroxy-2-({2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}methyl)quinoline-6-carboxamide
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-1-(piperidin-1-yl)propan-1-one
(3R,4R)-1-[2-(3-fluorophenyl)ethyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-(pyrrolidin-1-yl)butan-1-one
2-(benzyloxy)-1-(3-{[2-(dimethylamino)ethyl](methyl)amino}piperidin-1-yl)ethan-1-one
3-(3-chlorophenyl)-3-phenyl-N-(pyrimidin-4-ylmethyl)propanamide
N-methyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
(1S,5R)-3-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3,5-dimethyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1H-indole-2-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylbenzamide
N-(2-oxo-2-{2-[5-(thiomorpholine-4-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}ethyl)acetamide
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]propanamide
4-benzoyl-1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidine
(3aS,6aR)-3-[2-(pyridin-2-yl)ethyl]-5-(pyrimidin-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(2R,3S,6R)-5-(2-methyl-1,3-thiazole-4-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[1-(4-aminopyrimidin-2-yl)piperidin-4-yl]pyrrolidin-2-one
1-(3-ethyl-1H-pyrazole-4-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
N-[2-(benzyloxy)ethyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]piperazine
2-[2-(3-methoxyphenyl)piperidine-1-carbonyl]benzonitrile
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(thiophene-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]acetamide
(4aR,8aR)-2-methanesulfonyl-7-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-decahydro-2,7-naphthyridin-4a-ol
(1S,2R)-N1,N2-dimethyl-N1-(quinolin-5-ylmethyl)cyclohexane-1,2-dicarboxamide
1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one