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4-{[2-(3-methoxyphenyl)ethyl]amino}-N-(1-methoxypropan-2-yl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]pyrimidin-2-amine
5-[(4-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1,3-oxazol-2-yl)methoxy]isoquinoline
1-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]isoquinoline
2-{3-[1-(1,2,3,4-tetrahydronaphthalen-2-yl)-1H-imidazol-2-yl]phenoxy}acetamide
2-(1,3-benzoxazol-2-yl)-N-[2-(1-hydroxycyclopentyl)ethyl]-N-methylacetamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(quinoxalin-2-yl)pyrrolidin-3-yl]methanol
6-methyl-4-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-2-(pyrimidin-5-yl)quinoline
1-ethyl-N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-({4-[benzyl(methyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}methyl)benzonitrile
N-(2-methoxyethyl)-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2-cyclopropyl-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1,3-benzoxazole-6-carboxamide
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-2-(ethylsulfanyl)propan-1-one
3-phenyl-1-(9H-purin-6-yl)pyrrolidin-3-ol
N'-methyl-N'-[(4-phenoxyphenyl)methyl]butanediamide
3-(2-methylpropyl)-N-(2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1H-pyrazole-5-carboxamide
(3aS,7aR)-2-(2-{[(4-fluorophenyl)methyl](methyl)amino}acetyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-cyclopentanecarbonyl-N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
N-(3-methoxypropyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]acetamide
N-[(2-methoxyphenyl)methyl]-N-{[1-(propan-2-yl)piperidin-4-yl]methyl}cyclopropanamine
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
3-[2-(dimethylamino)ethyl]-5-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-5-(3-methylbutyl)imidazolidine-2,4-dione
5-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}pyrrolidin-2-yl)-3-phenyl-1,2,4-oxadiazole
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-1,3-benzothiazole-2-carboxamide
(1R,5R)-3-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
3,5-dimethyl-N-(pyrimidin-4-ylmethyl)-1-benzofuran-2-carboxamide
1-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methyl-3-(1H-1,2,4-triazol-1-yl)propan-1-one
(3S,4S)-1-[(5-chloro-2-hydroxyphenyl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
4-ethyl-3-{[1-(quinolin-2-ylmethyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-(3-phenyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-amine
2-[3,5-dimethyl-4-(quinolin-6-yl)-1H-pyrazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
[(3R,4S)-1-[(4-tert-butylphenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
4-methyl-9-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
(3R,4S)-4-cyclopropyl-1-[5-(ethylsulfanyl)thiophene-2-carbonyl]pyrrolidin-3-amine
N-methyl-2-(phenylamino)-N-[1-(pyridin-3-yl)pentyl]pyrimidine-5-carboxamide
N-methyl-N-[(5-{[3-(3-methylphenoxy)azetidin-1-yl]methyl}furan-2-yl)methyl]methanesulfonamide
(2S,4R)-4-(3-fluorobenzamido)-N-methyl-N-[2-(pyridin-2-yl)ethyl]pyrrolidine-2-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2,8-dimethylquinoline-4-carboxamide
1-[3-(3-hydroxy-3-methylbutyl)benzoyl]-4-(pyridin-3-yl)piperidin-4-ol
5-fluoro-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]quinazolin-4-amine
(3R)-1-[(3,5-dichloropyridin-4-yl)methyl]-3,4,4-trimethylpyrrolidin-3-ol
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-methylpyrazin-2-amine
N-{2-[2-(methylcarbamoyl)ethyl]phenyl}-3-(2-methylpiperidin-1-yl)azetidine-1-carboxamide
(2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}-2-oxoethyl)urea
5-(phenoxymethyl)-N-[2-(1,3-thiazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
[(3R,4R)-1-[(3,5-dimethyl-1H-indol-2-yl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
8-[3-(1,3-benzothiazol-2-yl)propanoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one