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1,5-dimethyl-3-{[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-1H-indazole
(3S,4S)-1-(5-methylthiophene-3-carbonyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
4-phenyl-5-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-1,3-thiazole
4-(4-chloro-2-fluorobenzoyl)-1-(3-chlorophenyl)-5-methylpiperazin-2-one
3-[6-amino-5-cyano-4-(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)pyridin-2-yl]-1H-pyrazole-5-carboxylic acid
(4aR,7aS)-1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3aR,6aR)-2-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-chloro-6-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]pyridine-2-carboxylic acid
[1-(1-{[4-(pyridin-2-yl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanol
1-[(2E)-3-phenylprop-2-en-1-yl]-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperazine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-methylpyrrolidin-3-yl]-3,4,7-trimethyl-1H-indole-2-carboxamide
1-[(2-fluorophenyl)methyl]-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-6-oxopiperidine-3-carboxamide
N-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-N-methyl-1H-pyrazole-4-carboxamide
1-[3-(1H-imidazol-2-yl)benzoyl]-2-(3-methoxyphenyl)piperidine
(5-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
benzyl({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
4-{1-[3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}benzoic acid
3-(8-methoxyquinolin-5-yl)-4H-chromen-4-one
3-[5-(1H-pyrrole-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
N-cyclohexyl-5-[1-(3-hydroxypyridine-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
3,5-dimethyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1-benzofuran-2-carboxamide
(2,1,3-benzothiadiazol-5-ylmethyl)({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
2-({2-[1-(5-propyl-1,3,4-thiadiazol-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-2-(thiophen-3-yl)acetamide
1-[(2-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3,5-dimethyl-N-{3-methyl-1-[7-(3-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}benzamide
6-ethyl-2-(morpholin-4-yl)-N-(1H-1,2,4-triazol-5-ylmethyl)pyrimidin-4-amine
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-1-propyl-1H-pyrazole-5-carboxamide
1-[2-(pyridin-4-yl)-4-[(1H-1,2,4-triazol-3-ylmethyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-methoxy-2-phenylacetamide
6-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-1H-indole
4-{[2-(2-fluorophenyl)ethyl]amino}-N-(furan-2-ylmethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-[5-(2,3-dimethylphenyl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
3-(2-fluorophenyl)-1-(2-methoxyethyl)-3-{2-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
N-methyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-7H-pyrrolo[2,3-d]pyrimidin-4-amine
4-chloro-N,N-dimethyl-5-[(2-phenylmorpholin-4-yl)methyl]-1,3-thiazol-2-amine
9-[3-(methylsulfanyl)propanoyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
6-(propan-2-yl)-N4-[1-(pyrimidin-4-yl)ethyl]pyrimidine-2,4-diamine
5-(3-methoxyphenoxymethyl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-pyrazole-3-carboxamide
methyl N-{4-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]phenyl}carbamate
N-cyclopropyl-N-({3-[(2-fluorophenyl)methoxy]phenyl}methyl)thiophene-2-carboxamide
1-{2,7-diazaspiro[4.5]decan-2-yl}-4-(4-methoxyphenyl)butan-1-one
(4aS,7aR)-1-[3-(3-methoxy-4-methylphenyl)propanoyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-{1-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
N-methyl-N-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}oxan-4-amine
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]piperidine
[1-(2,5-dimethylpyrimidin-4-yl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1-[4-(4-methyl-1H-pyrazol-3-yl)piperidin-1-yl]ethan-1-one
methyl({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)(quinolin-4-ylmethyl)amine