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(3S,4S)-1-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-4-(naphthalen-2-yl)piperidin-3-ol
4-[3-({1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}oxy)benzoyl]morpholine
methyl 4-[(3-{[2-(4-methoxyphenyl)acetamido]methyl}piperidin-1-yl)methyl]benzoate
3-ethyl-8-[2-(5-ethyl-1-benzofuran-3-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-methyl-1-{8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}pyrrolidine-3-carboxamide
N-(2-methoxyethyl)-1-[1-(1-methyl-1H-imidazole-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
1-[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)ethan-1-one
N-{2-[(2-chlorophenyl)formamido]ethyl}-3-(1-methylpiperidin-2-yl)propanamide
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(naphthalene-2-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(2-chloro-4-fluorophenoxymethyl)-N-[(3S)-2-oxoazepan-3-yl]-1,3-oxazole-4-carboxamide
N,N-dimethyl-2-{[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}benzenesulfonamide
(1S,5R)-N-(6-chloropyridin-3-yl)-10-oxo-3,9-diazabicyclo[3.3.2]decane-3-carboxamide
5-(methanesulfonylmethyl)-2-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]pyridine
(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)urea
4-{[(4aS,7aR)-4-[2-(dimethylamino)acetyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
1-(2-fluorophenyl)-4-{[4-(3-methoxypiperidine-1-carbonyl)-1,3-oxazol-2-yl]methyl}piperazine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)acetamide
ethyl 5-(1H-1,3-benzodiazol-2-ylmethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,3,6-trimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
2-(azepan-1-yl)-2-oxo-N-[2-(4-propylmorpholin-2-yl)ethyl]acetamide
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-[(3-ethoxy-4-methoxyphenyl)methyl]-N-methyl-3-(4H-1,2,4-triazol-4-yl)benzamide
3-[1-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)piperidin-2-yl]propan-1-ol
1-(2-methylpropyl)-5-oxo-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidine-3-carboxamide
6-(6-methoxypyridin-3-yl)-N,N-dimethylpyridine-2-carboxamide
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-{[4-(trifluoromethyl)phenyl]methyl}acetamide
2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5-(trifluoromethyl)pyridine
dimethyl({2-[2-(1-phenylmethanesulfonylpiperidin-4-yl)-1H-imidazol-1-yl]ethyl})amine
1-(4-{[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}piperidin-1-yl)ethan-1-one
(2E)-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-hydroxyethan-1-one
3-[5-(pent-2-yn-1-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
2-{[4-(2-methoxy-5-methylphenyl)-5-(1-methoxyethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-(2-hydroxyphenoxy)ethan-1-one
methyl({[3-(methylsulfanyl)phenyl]methyl})(piperidin-4-ylmethyl)amine
[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl})amine
1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}ethan-1-one
1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
N-[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
[3-(3-methoxypropyl)-1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]methanol
(3S,9R)-11-(2,4,5-trifluorobenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
(2S)-2-(methoxymethyl)-N-[3-(1,3-oxazol-5-yl)phenyl]pyrrolidine-1-carboxamide
methyl 1-(2-methoxyethyl)-5-{[(5-methylfuran-2-yl)methyl]amino}-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(3-hydroxyquinoxalin-2-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]propanamide
3-(ethoxymethyl)-1-(2-methylphenyl)-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazole
6-methyl-5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]imidazo[2,1-b][1,3]thiazole
1-(4-aminopyrimidin-2-yl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylic acid
5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-N-methylpyrimidin-2-amine
(4aR,8aR)-4-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-octahydro-2H-1,4-benzoxazine