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5-{[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]methyl}-2-methoxyphenol
N-{[(3S,4S)-1-(2-cyanobenzoyl)-3-hydroxypiperidin-4-yl]methyl}-2-cyclopentylacetamide
(3S,4S)-4-(morpholin-4-yl)-1-[1-(4-phenylphenyl)-1H-1,2,3,4-tetrazol-5-yl]pyrrolidin-3-ol
5-{[2-(3-methoxyphenyl)ethyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-[2-(2,6-difluorophenyl)acetyl]-1-(2-methylphenyl)piperazin-2-one
4-(2-methylphenyl)-3-[1-(1H-pyrazol-1-yl)ethyl]-4H-1,2,4-triazole
1-(2,3-dihydro-1H-inden-2-yl)-4-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
2-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[4-(2,2-dimethyloxan-4-yl)-1H-1,2,3-triazol-1-yl]-N-(2,4-dimethylphenyl)propanamide
4-[(2-chlorophenyl)methyl]-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{1-[1-(2-methoxy-2-phenylacetyl)piperidin-4-yl]-2-phenylethyl}-N,2-dimethylfuran-3-carboxamide
1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(1H-1,2,3-triazol-1-yl)ethan-1-one
methyl 2-({[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(methyl)amino)acetate
3-methyl-6-[4-(3-methylpyridin-2-yl)piperazin-1-yl]pyridazine
[(4aS,8aR)-6-[(5-chlorothiophen-2-yl)sulfonyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
5-(propan-2-yl)-4-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}pyrimidine
N-{1-[1-(4-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]piperidin-4-yl}pyridin-2-amine
N4-[(1R,3R)-3-aminocyclopentyl]-2-(butylsulfanyl)pyrimidine-4,6-diamine
2,2-dimethyl-6-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-3,4-dihydro-2H-pyran-4-one
2-{3-[2-(2,4-difluorophenyl)ethyl]piperidine-1-carbonyl}pyridine
[(1R,3S,3aS,6aR)-3-(4-butoxyphenyl)-1,5-dimethyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
6-chloro-2-{[1-(2-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
2-{2-[(2,2-dimethylmorpholin-4-yl)methyl]-4-(4-fluorophenyl)phenoxy}acetic acid
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
(3R,4R)-4-amino-1-[2-(2-methoxy-4-methylphenoxy)ethyl]piperidin-3-ol
(3aR,6aR)-2-(prop-2-en-1-yl)-5-(4,4,4-trifluorobutanoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(carbamoylmethoxy)-N-methyl-N-(prop-2-yn-1-yl)benzamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(3R,4S)-1-cyclopentyl-4-(propan-2-yl)pyrrolidin-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
N-[(3R,4R)-1-[2-(2,3-dimethylphenoxy)acetyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
1-[2-amino-4-(cyclopropylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-4-(1H-imidazol-1-yl)butan-1-one
1-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(1H-pyrazol-1-yl)propan-1-one
5-[3-(furan-2-yl)phenyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-{2-[(2-methoxyphenyl)methyl]pyrimidin-4-yl}pyridine-4-carboxylic acid
1-(5-methoxyfuran-2-carbonyl)-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine
[(3R,4R)-1-(8-fluoroquinoline-2-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]azepane
2-ethyl-4-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-2-(2,5-dimethoxyphenyl)-N-methylacetamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[(2E)-3-phenylprop-2-enoyl]-decahydro-1,6-naphthyridin-2-one
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(cyclopropylmethyl)acetamide
4-{3-cyclopentyl-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl}benzene-1-sulfonamide
N-cyclopropyl-3-[5-(pyridine-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
1-methyl-N-(2,2,2-trifluoroethyl)-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
{5-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]furan-2-yl}methanol
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]pyrimidine-5-carboxamide
N-(1-benzylpiperidin-3-yl)-5-phenyl-1,2,4-triazin-3-amine
{1-[5-(2,5-dimethylfuran-3-yl)-1,2,4-triazin-3-yl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(ethanesulfonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane