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1-{9-[2-(2-methoxyethyl)morpholin-4-yl]-3-azaspiro[5.5]undecan-3-yl}-2-methylpropan-1-one
3-ethyl-1-methyl-6-(pyridin-3-ylmethyl)-1H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
2-[5-(1H-imidazol-4-ylmethyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]-1H-1,3-benzodiazole
(1R,3S)-3-(2-hydroxyethoxy)-7-{pyrazolo[1,5-a]pyridine-3-carbonyl}-7-azaspiro[3.5]nonan-1-ol
N-[(2S)-1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-1-oxopropan-2-yl]acetamide
5-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
[(2-methoxyphenyl)methyl][(1-methyl-1H-imidazol-2-yl)methyl](pyridin-3-ylmethyl)amine
N-(1,2-oxazol-3-ylmethyl)-3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
[3-(1H-imidazol-4-ylmethyl)-9-[3-(1H-pyrazol-1-yl)propyl]-3,9-diazaspiro[5.5]undecan-1-yl]methanol
ethyl 4-(3-phenylpropyl)-1-[3-(pyrazin-2-yl)propanoyl]piperidine-4-carboxylate
2-(3-{3-[6-(dimethylamino)pyridazin-3-yl]phenyl}-1H-pyrazol-1-yl)-N-(furan-2-ylmethyl)acetamide
7-(4-aminopyrimidin-2-yl)-N4-(1,2-oxazol-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
(4aS,7aR)-1-(2-methylfuran-3-carbonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-methoxy-6-methylphenyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecane-11-carboxamide
3-(5-methylfuran-2-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-pyrazole-5-carboxamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(morpholin-3-yl)acetamide
N,6,6-trimethyl-5-oxo-N-[(4-phenylphenyl)methyl]thiomorpholine-3-carboxamide
N-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)propanamide
N-(1H-imidazol-4-ylmethyl)-N-(pyridin-3-ylmethyl)cycloheptanamine
4,6-dimethyl-1-[2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,2-dihydropyrimidin-2-one
2-{4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
1-[(1-{6-[(3-hydroxypropyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
(3S)-3-(dimethylamino)-N-{4-[ethyl(phenyl)carbamoyl]phenyl}pyrrolidine-1-carboxamide
6-[(3R,4R)-3-[(4-ethylpiperazin-1-yl)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]pyridine-2-carbonitrile
2-{4-[(dimethylamino)methyl]phenoxy}pyridine-3-carbonitrile
4-{5-fluoro-2-[2-(propan-2-yloxy)phenyl]pyrimidin-4-yl}morpholine
methyl (2S)-1-({4-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)pyrrolidine-2-carboxylate
2,4-dichloro-3-{[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]methyl}phenol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-oxobutanamide
2-[(2-fluorophenyl)methyl]-1,6-dimethyl-3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,4-dihydropyridin-4-one
8-(1H-imidazol-2-ylmethyl)-3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(2-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
N-cyclopropyl-4-methoxy-3-({[1-(thiophen-3-yl)propan-2-yl]carbamoyl}amino)benzamide
1-[4-(pyrazin-2-yl)piperazin-1-yl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
1-methyl-4-({5-[4-(1H-pyrrol-1-yl)phenyl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
2-{[2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]amino}-6-methyl-3,4-dihydropyrimidin-4-one
(4aR,7aS)-1-cyclopropanecarbonyl-4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]acetamide
(2R,3R,6R)-5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-methyl-4-{5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}-2-phenylpiperazine
4-{2-[1-(4,6-dimethylpyridine-3-carbonyl)piperidin-2-yl]ethyl}phenol
N-[(2-methoxyphenyl)methyl]-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-4'-yl}acetamide
2-(2,4-dimethoxy-3-methylphenyl)-1H-imidazole
7,7-dimethyl-2-[(1-methylpyrrolidin-2-yl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[(2-methylpyrimidin-5-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)imidazo[1,2-a]pyrimidine-2-carboxamide
2-amino-6-(4-methoxyphenyl)-5-methyl-4-(2-methyl-1H-imidazol-4-yl)pyridine-3-carbonitrile
N-(1-{4-[(2,2-diphenylethyl)carbamoyl]phenyl}-1H-pyrazol-4-yl)oxane-4-carboxamide
2-{[(3-cyanophenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide