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(1R,7S)-3-(2-ethylbutyl)-N-(furan-3-ylmethyl)-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-methyl-1-(oxolan-2-ylmethyl)-N-(pyrimidin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N4-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-(pyrrolidin-1-yl)pyrimidine-4,6-diamine
1-[4-(dimethylamino)azepan-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
5-methoxy-2-({3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}methyl)-4H-pyran-4-one
methyl (2R)-2-{[2-(phenoxymethyl)-1,3-oxazol-4-yl]formamido}propanoate
N-(4-{5-[(2-hydroxy-5-methylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)acetamide
ethyl 4-{2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamido}piperidine-1-carboxylate
1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
2-(4-{[4-(piperidin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}-1,3-thiazol-2-yl)pyrimidine
1-(5-chloro-2-hydroxy-3-{4-[1-(morpholin-4-yl)ethyl]phenyl}phenyl)ethan-1-one
6-methoxy-3-[(3-propoxypiperidin-1-yl)methyl]-1,2-dihydroquinolin-2-one
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[(2R)-1-hydroxy-3-phenylpropan-2-yl]benzamide
3-[7-(3-methoxypropyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]benzonitrile
(1S,5R)-6-(2-methoxyethyl)-3-[2-(1H-1,2,4-triazol-3-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
[(1-cyclohexylpiperidin-3-yl)methyl][(1-methyl-1H-pyrazol-4-yl)methyl](pyridin-3-ylmethyl)amine
(1S,5R)-3-[2-(methylamino)pyrimidine-5-carbonyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[4-(cyclopropylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
5-{[2-(4-fluorophenyl)piperidin-1-yl]methyl}-N,N-dimethylfuran-2-carboxamide
7-[(3S,4S)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-{6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-4-(4-ethyl-1H-pyrazol-5-yl)piperidine
(2S,4S)-4-(4-{2-[(3-methoxyphenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)acetamide
1-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
3-chloro-N-ethyl-4-fluoro-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-1-benzothiophene-2-carboxamide
2-chloro-N-{2-[(5-cyclobutyl-1,3,4-oxadiazol-2-yl)amino]ethyl}benzamide
N-methyl-4-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)benzene-1-sulfonamide
4-({6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1-methyl-1H-pyrrole-2-carbonitrile
2-cyclopentyl-N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
1-(4-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-3,5-dimethyl-1H-pyrrol-2-yl)ethan-1-one
2-(dimethylamino)-2-(4-fluorophenyl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)acetamide
1-(2-{4-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)piperazine
N-(1H-imidazol-2-ylmethyl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-[3-(1H-1,2,3-triazol-1-yl)propyl]urea
2-{2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-4-carboxamide
3-{[1-(carbamoylmethyl)pyrrolidin-3-yl]methyl}benzamide
N-[2-methyl-1-(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]methanesulfonamide
2-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1-benzofuran-5-carboxamide
N-(oxan-4-ylmethyl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
8-[(2,6-difluorophenyl)methyl]-2-phenyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
6-(5-ethoxyfuran-2-carbonyl)-2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
5-cyclopropyl-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1,3,4-oxadiazol-2-amine
1-(cyclopropanesulfonyl)-2-(4-fluorophenyl)piperidine
methyl (2S,4S)-1-methyl-4-(2-oxo-2H-chromene-6-sulfonamido)pyrrolidine-2-carboxylate
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N,3,5,7-tetramethyl-1H-indole-2-carboxamide
[(5-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}furan-2-yl)methyl]dimethylamine
N-(5-methyl-2-pentanamidophenyl)-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-{1-oxaspiro[4.4]nonan-3-yl}pyrimidin-2-amine
1-(4-chloro-2-methoxybenzoyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane