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3-{5-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]thiophen-2-yl}prop-2-yn-1-ol
N-(1H-1,3-benzodiazol-5-yl)-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(2S)-N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-5-oxopyrrolidine-2-carboxamide
N-[3-({[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]carbamoyl}amino)-4-methylphenyl]cyclopentanecarboxamide
4-[1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]benzoic acid
N-[3-(oxolan-3-yl)propyl]-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
methyl (2S,4R)-4-[2-(4-fluorophenyl)acetamido]-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}pyrrolidine-2-carboxylate
1-[3-({[2-(dimethylamino)pyrimidin-5-yl]methyl}amino)phenyl]pyrrolidin-2-one
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-7-methyl-1-benzofuran-2-carboxamide
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-(3-methyl-1H-pyrazol-5-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-1,4-diazepan-6-ol
5-methanesulfonyl-2-methyl-4-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]pyrimidine
2,4-dimethyl-5-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrimidine
5-methoxy-2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1H-indole
(3S,5S)-5-(3,3-diphenylpiperidine-1-carbonyl)-1-methylpyrrolidin-3-amine
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}imidazo[1,2-a]pyridine-3-carboxamide
1-(2-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)piperidin-2-one
N3-(butan-2-yl)-1-cyclopentyl-N5-(3-ethoxypropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-{1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-1H-pyrazole-4-carbonyl}morpholine
6-methyl-3-[1-(pyridin-2-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[3-(pyridin-4-yl)propyl]-1H-pyrazole-4-carboxamide
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-6-methylpyridine-2-carboxamide
1-(cyclopropylmethyl)-4-(1-methyl-1H-pyrazole-5-carbonyl)-2-(propan-2-yl)-1,4-diazepane
2-(1-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-1H-1,2,3-triazol-4-yl)benzoic acid
6-fluoro-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-{[3-(2,6-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-benzoxazole
1-(2-methyl-1,3-thiazole-5-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-2-(2-phenylethyl)piperidine
1-[6-(cyclopentylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-N,N-diethylpiperidine-4-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-(3-fluoro-4-methoxybenzenesulfonyl)pyrrolidine-2-carboxamide
4-{3,9-diazaspiro[5.6]dodecane-9-carbonyl}-N-(pyridin-4-ylmethyl)aniline
2-cyclohexyl-N-{[(3S,4S)-3-hydroxy-1-(oxane-4-carbonyl)piperidin-4-yl]methyl}acetamide
1-[(4-fluorophenyl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]-1,4-diazepane
2-methyl-4-(2-methylphenyl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperazine
N-(2-cyclopropylphenyl)-2-{3-[3-(pyrimidin-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
2-[3-(3-acetylphenyl)-1H-indazol-1-yl]-N-(1,3-dimethyl-1H-pyrazol-5-yl)acetamide
(2S)-2-amino-N-methyl-4-(methylsulfanyl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}butanamide
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]oxane-4-carboxamide
(2S)-2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetamido]-3-phenylpropanamide
[(2R)-1-({1-[1-(2-methylpyridin-4-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)pyrrolidin-2-yl]methanol
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}ethan-1-one
[(3R,4R)-1-(6,8-dimethylquinolin-4-yl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
4-[(4-fluorophenyl)methyl]-1-[(3-methylpyridin-2-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
4-[1-(2-methoxypyridine-4-carbonyl)piperidin-4-yl]-6-(pyrrolidin-1-yl)pyrimidine
N-(oxolan-3-yl)-3-[(pyridin-4-ylmethyl)sulfamoyl]benzamide
2-[4-({2-oxo-1-oxa-3,8-diazaspiro[4.6]undecan-8-yl}methyl)phenyl]acetic acid
{1-[({[4-(difluoromethoxy)phenyl]methyl}(methyl)amino)methyl]cyclopentyl}methanol
3-methoxy-1-{2-oxo-2-[4-(2-oxo-1,3-oxazolidin-3-yl)piperidin-1-yl]ethyl}-1,2-dihydropyridin-2-one
1-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-4-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide