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N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-(1,2-oxazolidin-2-yl)propanamide
1-{4-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]thiophen-2-yl}ethan-1-one
6-fluoro-2-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1H-1,3-benzodiazole
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-5-methyl-1,3-oxazole-4-carboxamide
N-(furan-2-ylmethyl)-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{2-methoxy-5-[({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}amino)methyl]phenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
5-{1-[4-(2-methoxynaphthalen-1-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
2-[(E)-2-phenylethenyl]-4-(3,3,3-trifluoropropyl)pyrimidine
(1S,3R)-3-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}cyclohexan-1-amine
[(1-cyclopentylpiperidin-4-yl)methyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
3-{2-[(4-methoxyphenyl)methyl]morpholin-4-yl}propanoic acid
1-[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-phenoxypropan-1-one
N,N-diethyl-1-[5-(4-methoxyphenyl)-1,2,4-triazin-3-yl]pyrrolidin-3-amine
methyl[(3-phenyl-1,2-oxazol-5-yl)methyl](pyridin-4-ylmethyl)amine
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]acetamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]propan-1-one
1-{1-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidin-4-yl}pyrrolidin-2-one
6-ethyl-N-[2-hydroxy-2-(4-hydroxyphenyl)ethyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
3-(2-ethyl-1H-1,3-benzodiazol-1-yl)-1-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]propan-1-one
4-[1-({1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]pyridine
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]benzamide
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]pyrrolidin-3-yl]urea
N-[2-(2-fluoro-5-methylphenyl)pyridin-3-yl]-2-methylpropanamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1H-pyrazole-3-carboxamide
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(3-fluorophenyl)methyl]urea
1-(2-chlorophenyl)-3-[1-(1-cyclopropanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]urea
5-[4-(1-hydroxy-3-phenylpropyl)piperidine-1-carbonyl]pyrazin-2-ol
N-(1,3-benzoxazol-2-ylmethyl)-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-propanamido-N-[3-(pyridin-4-yl)propyl]benzamide
1-{1,3-dioxo-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}-N-(thiophen-3-ylmethyl)piperidine-3-carboxamide
methyl 3-(2-methoxyacetamido)-1-[2-(4-methoxyphenyl)ethyl]-5-[(thian-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-{4-[(4-fluorophenyl)methyl]-6-hydroxy-1,4-diazepane-1-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
1-[2-(2-fluoro-6-methoxyphenyl)pyridine-4-carbonyl]-4-methylpiperazine
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl}propanamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
3-(4-{[methyl(oxan-4-ylmethyl)amino]methyl}-1H-pyrazol-1-yl)propanoic acid
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](2-methoxyethyl)[(4-methylphenyl)methyl]amine
N-[2-(furan-2-yl)ethyl]-1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]piperidin-4-amine
4-hydroxy-3-methyl-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]benzamide
N-[(5-chloro-1H-indol-2-yl)methyl]-2-(3-hydroxyphenyl)acetamide
N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-2-(pyridin-2-yl)acetamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
3-[(4S)-2,5-dioxoimidazolidin-4-yl]-N-[3-(pyridin-3-yl)propyl]propanamide
4-{[(1R,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzoic acid
N-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)thiomorpholine-4-carboxamide
1-[(2-fluorophenyl)methyl]-N-methyl-N-[(4-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]-3-(hydroxymethyl)morpholine-4-carboxamide
N,N-diethyl-2-(4-{4-[(3-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-1H-1,2,3-triazol-1-yl)acetamide
N-ethyl-5-[(3-phenylpiperidin-1-yl)methyl]pyrimidin-2-amine
1-(furan-3-ylmethyl)-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide