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N,N-diethyl-1-{5-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}pyrrolidin-3-amine
4-cyclobutanecarbonyl-N-(3,4-dimethylphenyl)-1,4-diazepane-1-carboxamide
methyl 5-{[(3-fluorophenyl)methyl]amino}-3-(4-methoxybenzamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[2-(pyrrolidin-1-yl)ethyl]-1,3-oxazole-4-carboxamide
N-ethyl-N-(2-hydroxyethyl)-2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
5-(3,4-difluorophenoxymethyl)-N-[2-(methylsulfanyl)ethyl]-1,2-oxazole-3-carboxamide
1-{4-[2-(cyclopentylmethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}-2-(3-fluorophenyl)ethan-1-one
2-(2,6-dichlorophenyl)-1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]ethan-1-one
2-methyl-6-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
[(3-methylthiophen-2-yl)methyl]({[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl})(pyridin-2-ylmethyl)amine
3-(1-{1-azabicyclo[2.2.2]octan-3-yl}-4-phenyl-1H-imidazol-5-yl)quinoline
2-methyl-6-(1-{[4-(pyridin-2-yl)phenyl]methyl}piperidin-3-yl)pyrimidin-4-ol
1-({4-methyl-5-[1-(pyrazin-2-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
1-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazol-2-yl)piperidine
(2S,4R)-4-cyclopentaneamido-N,N-diethyl-1-[(4-methyl-1H-imidazol-2-yl)methyl]pyrrolidine-2-carboxamide
1-cyclobutanecarbonyl-N-{[3-(methylcarbamoyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carboxamide
(4aS,7aR)-N-[2-(4-methoxyphenyl)ethyl]-4-methyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
7-[4-(2-fluorophenyl)piperazine-1-carbonyl]-2-(2-methoxyphenyl)-1-methyl-1H-1,3-benzodiazol-5-amine
N-[3-(1H-indol-1-yl)propyl]-1,9-dioxaspiro[5.5]undecan-4-amine
1-(2-chlorophenyl)-4-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
(3R,9aR)-8-(4-chlorobenzenesulfonyl)-3-(hydroxymethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
8-methyl-3-{[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methyl}-1,2-dihydroquinolin-2-one
4-benzyl-3-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-(2-methylprop-2-en-1-yl)acetamide
methyl 2-[(butan-2-yl)sulfamoyl]-6-{[2-(trifluoromethyl)phenyl]methyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-[3-(4-ethylphenyl)-1H-pyrazole-5-carbonyl]-1-phenylpiperazin-2-one
4-[5-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
(2S,4R)-4-amino-1-(5-chloro-2-methoxybenzoyl)-N-ethylpyrrolidine-2-carboxamide
4-fluoro-2-{[methyl({[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}phenol
(3R,4S)-4-[methyl({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amino]oxolan-3-ol
5-cyclopropyl-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,3,4-oxadiazol-2-amine
2-[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]-5-fluoro-1H-1,3-benzodiazole
2-(2H-1,3-benzodioxol-5-yl)-4,6-dimethylpyridine-3-carbonitrile
(1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-4-(3-phenylpropyl)piperidin-4-yl)methanol
1-cyclohexyl-3-(cyclopropylmethyl)-N-(2,2-difluoroethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N-(4-methoxyphenyl)-1-methylpyrrolidine-3-carboxamide
(1R,5R)-6-benzyl-3-(3-chloro-4-fluorobenzoyl)-3,6-diazabicyclo[3.2.2]nonane
(4aR,7aS)-1-methanesulfonyl-4-(3-methyl-1,2-oxazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3-methoxyphenyl)methyl]-N,1-dimethyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[3-(4-fluorophenyl)phenyl]-1-(4-methyl-1,3-oxazole-5-carbonyl)pyrrolidine-2-carboxamide
N-cyclopentyl-7-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
8-[(4-hydroxyphenyl)methyl]-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4R)-1-[(4-chlorophenyl)methyl]-N,N-diethyl-4-[(1-methylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
1-[7-(3-chlorophenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-{[1-(oxolane-3-carbonyl)piperidin-4-yl]oxy}-N-(pyridin-3-ylmethyl)benzamide
N-(1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
2-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}benzonitrile