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methyl(pyrimidin-2-ylmethyl)[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-[(2-methoxyethyl)amino]pyridine-3-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-(1,5-dimethyl-1H-pyrazol-4-yl)-1H-pyrazole-3-carboxamide
6-(2-fluorophenyl)-N-methyl-N-[1-(pyridin-3-yl)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(4-fluorophenyl)-4-[2-(2-hydroxyethoxy)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{2-[cyclopentyl(methyl)amino]ethyl}-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1-propylpiperidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
4-fluoro-N-[(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)methyl]benzamide
N-[(1S,6R)-6-carbamoylcyclohex-3-en-1-yl]-4-[(diethylamino)methyl]-5-ethylfuran-2-carboxamide
(1S,5R)-6-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-cyclohexylpiperazin-2-yl}ethan-1-ol
1-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}isoquinoline
1-[1-(2-ethylpyrimidine-5-carbonyl)piperidin-4-yl]-3-methylbutan-1-ol
N-(dicyclopropylmethyl)-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
2-(2-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}phenoxy)acetic acid
{2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}urea
methyl 5-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
2-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-2,3-dihydro-1H-isoindole
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-[(3-methoxyphenyl)methyl]-N-methylpropanamide
5-(1-benzofuran-2-yl)-N-methyl-N-(pyridin-3-ylmethyl)-1,2,4-triazin-3-amine
2-[4-(2,6-dimethoxypyrimidin-4-yl)-1-methylpiperazin-2-yl]ethan-1-ol
N2-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-N1-(3-methylpyridin-2-yl)ethane-1,2-diamine
(2S,4R)-4-[(naphthalen-2-ylmethyl)amino]-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
{4-[5-(methanesulfonylmethyl)pyridin-2-yl]phenyl}methanol
6-fluoro-2-({[3-(pyridin-3-yloxy)propyl]amino}methyl)quinolin-4-ol
9-oxo-N-(prop-2-en-1-yl)-N-(propan-2-yl)-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
ethyl 2-{3-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)pyridin-4-yl]pyrrolidin-1-yl}acetate
3-(2H-1,3-benzodioxol-5-yl)-N-[1-(pyrazin-2-yl)piperidin-3-yl]propanamide
1-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(methylsulfanyl)ethan-1-one
N-(3-chloro-2-fluorophenyl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carboxamide
[7-(2H-1,3-benzodioxol-5-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methanamine
(2R,3R,6R)-3-phenyl-5-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
N,N-dimethyl-3-[methyl(oxan-4-yl)sulfamoyl]benzamide
dimethyl[2-(2-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]amine
1-[2-(3-phenylpropyl)morpholin-4-yl]-2-(pyridin-3-yl)ethan-1-one
5-{4-phenyl-1-[1-(pyrazin-2-yl)propan-2-yl]-1H-imidazol-5-yl}-2,1,3-benzoxadiazole
2-methoxy-5-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}benzoic acid
1,3-dimethyl-N-[2-(4-methyl-1H-pyrazol-1-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
[(2,4-dimethoxyphenyl)methyl](methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]-1-methyl-1,4-dihydroquinolin-4-one
2-amino-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)pyridine-4-carboxamide
2-ethyl-4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholine
N,2-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-[(pyridin-2-ylmethyl)amino]benzamide
4-{[5-(oxolane-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}thiomorpholine
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({[3-(morpholin-4-yl)propyl]amino}methyl)phenoxy]propan-2-ol
1-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
1-(3-chlorophenyl)-3-[1-(1,1-dioxo-1λ6-thian-4-yl)piperidin-4-yl]urea
N-[2-(1H-indol-1-yl)ethyl]-N,2-dimethyl-1,3-thiazole-4-carboxamide