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({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl){[4-(pyrimidin-2-yloxy)phenyl]methyl}amine
1-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
4-[1-(4-methoxyphenyl)cyclopropanecarbonyl]piperazine-2-carboxylic acid
4-{[3-hydroxy-1-(2-methoxyethyl)-2-oxopiperidin-3-yl]methyl}-1-methylpiperazin-2-one
5-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
methyl 1-[(3S,5S)-5-(cycloheptylcarbamoyl)-1-[(3-methoxyphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
5-fluoro-2-(5-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)-1H-1,3-benzodiazole
(2S)-N2-[2-(2-methoxyphenyl)ethyl]pyrrolidine-1,2-dicarboxamide
N-[(2S)-1-methoxypropan-2-yl]-3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)benzene-1-sulfonamide
3-({[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}(methyl)amino)-1λ6-thiolane-1,1-dione
2-[4-(hydroxymethyl)phenyl]-2-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}acetic acid
5-[ethyl(2-methylprop-2-en-1-yl)amino]-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3S,9aR)-3-(4-aminobutyl)-8-(cyclopropylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[5-(1-ethyl-1H-indol-5-yl)-4-phenyl-1H-imidazol-1-yl]propanamide
N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]acetamide
N-{[1-(1,2-oxazol-3-ylmethyl)piperidin-3-yl]methyl}pyridine-3-carboxamide
6-[(3,5-dimethoxyphenyl)methoxy]-4-(3-phenyl-1,2-oxazole-5-carbonyl)-1-(propan-2-yl)-1,4-diazepan-2-one
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-yl)acetamide
1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-(oxolane-2-carbonyl)piperazine
(1S,5R)-3-[(1-methyl-1H-indol-6-yl)methyl]-3,9-diazabicyclo[3.3.2]decan-10-one
3-(4-cyclobutanecarbonyl-1,4-diazepane-1-carbonyl)-6-fluoroquinolin-4-ol
7-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}quinolin-8-ol
3-(4-chlorophenyl)-1-(4-methyl-1,4-diazepan-1-yl)-3-phenylpropan-1-one
N-(5-chloro-2-methoxyphenyl)-3-[1-(quinoline-6-carbonyl)piperidin-3-yl]propanamide
2-[3-({4-[(3,5-dimethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenoxy]ethan-1-ol
2-(3-hydroxypropyl)-9-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[(cyclohexylamino)methyl]-1-[(2-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
3-{5-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]thiophen-3-yl}prop-2-yn-1-ol
(3S,4R)-1-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-4-phenylpyrrolidine-3-carboxylic acid
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(propan-2-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
1-benzoyl-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
1-cyclobutanecarbonyl-4-[(2-fluoro-3-methoxyphenyl)methyl]-1,4-diazepane
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,5-thiadiazole-3-carboxamide
(3S,4S)-1-[(6-methylpyridin-2-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
N-benzyl-N,1-dimethyl-5-[(pyridin-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-propanamidobenzamide
1-ethyl-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]piperidine-2-carboxamide
2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-(3-hydroxy-3-phenylpyrrolidin-1-yl)ethan-1-one
3-(4-phenoxybenzoyl)-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine
1-(furan-2-ylmethyl)-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]piperidine-4-carboxamide
5-(methoxymethyl)-N-(oxan-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
methyl 3-benzamido-5-[(5-methylhex-5-en-2-yl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-cyclopropyl-N-[4-(morpholin-4-ylmethyl)phenyl]-1H-pyrazole-5-carboxamide
[3-({1-[(2-chloro-4-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)-2-[3-(trifluoromethyl)phenyl]acetamide
2-methyl-4-[2-(4-methylpentyl)morpholine-4-carbonyl]-1H-1,3-benzodiazole
1-[4-phenyl-1-(1,2,3,4-tetrahydroisoquinoline-6-carbonyl)piperidin-4-yl]ethan-1-one
1-[3-(5-methylfuran-2-yl)butyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-3-(piperidin-3-yl)benzamide