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N-[(2-chlorophenyl)methyl]-3-methyl-4-oxo-N-(prop-2-en-1-yl)-3,4-dihydroquinazoline-7-carboxamide
4-[4-(5-chloro-2-methoxybenzoyl)-2-oxopiperazin-1-yl]benzonitrile
3-methyl-6-{5-[5-(pyrrolidin-2-yl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl}pyridazine
2-methoxy-2-phenyl-N-(1-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(thiolan-3-yl)butanamide
N-[2-(7-{[4-(dimethylamino)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]cyclobutanecarboxamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1,5-dimethyl-1H-indole-2-carboxamide
(1S,5R)-3-(pyrrolidine-1-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methyl-N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-(morpholin-4-ylmethyl)piperidin-2-one
1-{1-[6-(4-methoxyphenyl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
3-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
2,6-dihydroxy-N-[1-(3-methylpyridin-2-yl)propan-2-yl]benzamide
2-{5-[1-(1,3-benzoxazol-2-ylsulfanyl)propyl]-1-(2-hydroxyethyl)-1H-1,2,4-triazol-3-yl}acetamide
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-[3-(5-methylfuran-2-yl)butyl]-6-azaspiro[2.5]octane-1-carboxamide
5-{pyrazolo[1,5-a]pyridin-7-yl}-2,3-dihydro-1H-inden-1-one
4-[3-({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)propyl]-1,3-thiazol-2-amine
1-(2-fluoroethyl)-3-[3-(4-methanesulfonylphenyl)phenyl]-1H-pyrazole
1-(4-methylphenyl)-4-(1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperazin-2-one
(1S,5R)-6-(3-fluoro-4-methylbenzoyl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3R,4R)-1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-3,4-dimethylpyrrolidin-3-ol
N-[1-(7-{[2-(furan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-methylpropanamide
2-[4-(2,4-dimethylpyrimidine-5-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
4-(2-methoxyacetyl)-1-phenylpiperazin-2-one
3-[1-(1H-1,3-benzodiazol-2-yl)-3-(methylsulfanyl)propyl]-1-(3-methyl-1,2,4-thiadiazol-5-yl)urea
N-[(4-chlorophenyl)methyl]-5-methyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-methylbenzamide
N-methyl-N-(quinoxalin-2-ylmethyl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2,2-dimethyl-N-[(4-sulfamoylphenyl)methyl]oxane-4-carboxamide
N-{3-[(dimethylsulfamoyl)amino]phenyl}-4-(2-methoxyethyl)piperazine-1-carboxamide
1-(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)azetidin-3-ol
2-[2-oxo-2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(6-methylpyridin-2-yl)methyl]acetamide
N-[1-({[(2-methyl-1,3-thiazol-4-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide
N-(2-fluoro-5-methylphenyl)-2-{4-[3-(pyridin-3-yl)propanoyl]morpholin-3-yl}acetamide
4-{3-[1-(2-methylpropyl)piperidin-4-yl]pyrrolidine-1-carbonyl}pyridazine
[(2-fluoro-5-methoxyphenyl)methyl]({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl})amine
(3S,4S)-4-cyclopropyl-1-(4-phenylbutanoyl)pyrrolidine-3-carboxylic acid
(3S,4R)-1-(1H-imidazol-2-ylmethyl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
2-{5-[2-(1,2-oxazolidin-2-yl)ethyl]-3-(2-phenylethyl)-1H-1,2,4-triazol-1-yl}pyridine
2-[4-(4-benzylpiperazine-1-carbonyl)-5-cyclopropyl-1H-pyrazol-1-yl]-4-(3-methoxyphenyl)pyrimidine
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}[(2-methoxyphenyl)methyl]methylamine
(4aS,8aR)-6-[2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(1-cyclohexyl-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-yl)ethan-1-ol
(4aS,8aR)-6-(4-methyl-1,3-oxazole-5-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1-cyclohexyl-3-(2-hydroxypyridin-3-yl)-1-[2-(1H-indol-3-yl)ethyl]urea
7-[(2-fluorophenyl)methyl]-2-{[5-(hydroxymethyl)furan-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-(2-methoxyethyl)-3,6-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-benzofuran-2-carboxamide
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide