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N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2-methyl-N-(pyridin-4-ylmethyl)-1,3-thiazole-4-carboxamide
4-(3-phenylpropyl)-1,3λ6,4-oxathiazinane-3,3-dione
6-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoxaline
N-(2-methyl-1H-1,3-benzodiazol-6-yl)-4-[2-(pyrrolidin-1-yl)ethyl]piperazine-1-carboxamide
(3R,5S)-N3-(4-fluorophenyl)-N5-[(4-methoxyphenyl)methyl]-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
(1-{1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
2-{4-[3-(cycloheptylcarbamoyl)propanamido]piperidin-1-yl}acetic acid
4-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidine-1-carbonyl}pyridin-1-ium-1-olate
4-(1H-1,3-benzodiazol-1-yl)-1-(6-methylquinolin-4-yl)piperidine-4-carboxylic acid
1-methyl-3-({[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amino}methyl)-1,2-dihydroquinolin-2-one
6-[1-(2-methyl-1-benzofuran-7-carbonyl)piperidin-4-yl]pyrimidin-4-ol
{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}(pyridin-4-ylmethyl)amine
N-[(4-cyanophenyl)methyl]-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
(3S,4R)-3-benzyl-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-methylpiperidin-4-ol
methyl (2S)-1-(2-{4-[4-({imidazo[1,2-a]pyridin-3-ylmethyl}amino)piperidin-1-yl]phenyl}acetyl)pyrrolidine-2-carboxylate
(4aS,8aR)-6-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
6-methyl-2-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)quinolin-4-ol
N-[(3-fluorophenyl)methyl]-N-(1-methoxypropan-2-yl)-1-methyl-1H-pyrazole-5-carboxamide
(4aS,8aS)-2-cyclobutanecarbonyl-7-(1-methyl-1H-pyrazole-4-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
1-(4-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)butan-1-ol
2-{[1-(4-fluorophenyl)cyclopropyl]formamido}-4-methanesulfonylbutanoic acid
[(3R,4R)-1-{5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
2-(8-methoxyquinolin-5-yl)-N-(prop-2-en-1-yl)pyridine-3-carboxamide
4-(2,1,3-benzothiadiazol-4-yl)-1-(pentan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazol-3-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(piperidine-1-carbonyl)pyridin-2-amine
(3aS,6aS)-2-cyclopentanecarbonyl-5-[2-(pyridin-3-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-benzyl-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3-ethyl-1,4-diazepan-5-one
methyl 9-[2-(2-fluorophenyl)ethoxy]-7-oxo-3-(5-oxopyrrolidine-3-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2R)-2-cyclohexyl-2-hydroxy-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
(2E)-N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-3-(3-fluorophenyl)-N-(pyridin-2-ylmethyl)prop-2-enamide
7-(2,6-dimethylquinoline-4-carbonyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
(1R,9aR)-1-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-octahydro-1H-quinolizin-1-ol
(1S,5R)-3-{2-[(2-methoxyethyl)amino]-1-methyl-1H-1,3-benzodiazole-5-carbonyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(morpholin-4-yl)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethan-1-one
2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
N-{3-methyl-1-[1-(pent-2-yn-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]butyl}acetamide
2-(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}thiophen-2-yl)pyrrolidine
1-(2,6-dimethylpyrimidine-4-carbonyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-5-methyl-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
1-(piperidin-3-ylmethyl)-N-(2,2,2-trifluoroethyl)-1H-1,2,3-triazole-4-carboxamide
5-(azepane-1-carbonyl)-N-[(5-fluoro-2-methylphenyl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
(3S,4S)-1-[(5-methylthiophen-2-yl)methyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
5-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]furan-2-carboxamide
ethyl 2-(N-methyl-1-{1-[3-(morpholin-4-yl)propyl]-6-oxopiperidin-3-yl}formamido)acetate
4-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N-methyl-1,3-thiazol-2-amine
N,N-dimethyl-1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]azepan-4-amine
3-(1-methanesulfonylpiperidin-4-yl)-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea