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5-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-[(phenylsulfanyl)methyl]pyrimidin-4-ol
2,2-dimethyl-6-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-3,4-dihydro-2H-pyran-4-one
{5-[({1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}amino)methyl]furan-2-yl}methanol
2-[9-(cyclopropanesulfonyl)-7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]acetamide
2-oxo-N-[2-(quinolin-8-yloxy)ethyl]-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}-N-[(2-methylphenyl)methyl]piperidine-1-carboxamide
2-(2-methoxyethyl)-9-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-2,9-diazaspiro[5.5]undecan-3-one
1,3-dimethyl-N-[2-methyl-1-(pyrrolidin-1-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-ethyl-4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
1-ethyl-8-[(4-hydroxyphenyl)methyl]-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{4-phenyl-5-[(1E)-1-phenylprop-1-en-2-yl]-1H-imidazol-1-yl}acetamide
1-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]urea
N-{[7-chloro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
4-chloro-3-({2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)-1-methyl-1H-indazole
1-methyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-1H-pyrazole-5-carboxamide
2-({methyl[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amino}methyl)-3,4-dihydroquinazolin-4-one
1-cyclopropyl-5-{[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
4-[4-(3-cyclohexylpropanoyl)piperazin-1-yl]-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}-3-(1-methylpiperidin-2-yl)propanamide
4-(2,3-difluoro-6-methoxybenzoyl)-1-[(3-methylphenyl)methyl]piperazin-2-one
4-{5-[(2-methyl-4-phenylpiperazin-1-yl)methyl]-1,3-thiazol-2-yl}morpholine
N-methyl-N-[2-(4-methylphenoxy)ethyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
5-methyl-4-[3-(propoxymethyl)pyrrolidine-1-carbonyl]-1-propyl-1H-pyrazole
(1S,5R)-6-[3-(furan-2-yl)benzoyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-{4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-ol
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
(1R,2S,4R)-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
N-butyl-5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-amine
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidine-1-carbonyl}cyclopropan-1-amine
4-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-(4-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
3-acetamido-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}butanamide
3-{[4-(3-chlorophenyl)-5-{[(cyclohexylmethyl)(methyl)amino]methyl}-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
2-({6-[2-(hydroxymethyl)phenyl]pyridazin-3-yl}(methyl)amino)ethan-1-ol
(3R,4R)-4-[(2-phenylquinolin-4-yl)amino]piperidin-3-ol
3-(4-methoxyphenyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
N-[4-(1H-pyrazol-5-yl)phenyl]-1-(pyridin-3-ylmethyl)piperidine-3-carboxamide
5,6,7-trimethoxy-3-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1,2-dihydroquinolin-2-one
2-{1-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-1H-imidazol-2-yl}-6-methylpyridine
2-amino-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-6-(propan-2-yl)pyrimidine-4-carboxamide
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-[2-(4-chlorophenyl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
[(2S)-1-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}pyrrolidin-2-yl]methanol
1-[(2S,4R)-1-[(3-fluorophenyl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
2-({[(3R,4R)-1-[(2-aminopyridin-3-yl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
3-methyl-5-[1-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)pyrrolidin-2-yl]-1H-1,2,4-triazole
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetic acid
2-[(4-propylpiperazin-1-yl)methyl]-4-(pyridin-2-yl)phenol