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1-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-4-(hydroxymethyl)piperidin-4-ol
1-methyl-5-(1-methyl-1H-indole-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-(1-cycloheptylpiperidin-3-yl)-2-(2-methoxyphenoxy)acetamide
2-ethoxy-5-(2-ethylpyrimidin-4-yl)benzoic acid
3-[({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}amino)methyl]piperidin-3-ol
6-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(4-methoxybenzoyl)piperazine
1-ethyl-3-(pyridin-2-ylmethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-[2-(2-methoxyethoxy)acetyl]-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-1-methylcyclopropane-1-carboxamide
(1R,7S)-N-methyl-3-[(3-methylphenyl)methyl]-N-(1,2-oxazol-3-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[2-(diethylamino)ethyl]-5-(propan-2-yl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-2-(1-ethylpiperidin-4-yl)acetamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
1-[5-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1-methyl-1H-pyrrol-3-yl]ethan-1-one
(4aS,7aR)-1-(benzenesulfonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N6-cyclopropyl-N4-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N4-methylpyrimidine-2,4,6-triamine
1-butyl-5-[5-(methoxymethyl)thiophen-2-yl]-3-methyl-1H-1,2,4-triazole
2-(2-methoxyethyl)-8-(6-methyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(2E)-N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(3,4-dimethoxyphenyl)prop-2-enamide
N-benzyl-N-methyl-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidin-3-amine
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-methylthiophene-2-carboxamide
2-[3-(4-methoxyphenyl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]benzonitrile
(3R,4R)-1-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-4-(morpholin-4-yl)piperidin-3-ol
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(4aS,8aR)-1-butyl-6-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carboxylic acid
(3S,4S)-1-(7-fluoro-3-methyl-1H-indole-2-carbonyl)-4-methylpiperidine-3,4-diol
3-({1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
2-(2-{[4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenoxy)acetamide
1-methyl-5-{[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}piperidin-2-one
N-(2-methoxyethyl)-N-[(2-methoxyphenyl)methyl]-1,3-dimethyl-1H-indole-2-carboxamide
6-fluoro-2-({4-[2-(pyrrolidin-1-yl)ethyl]piperazin-1-yl}methyl)quinolin-4-ol
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
8-(1-benzofuran-3-carbonyl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(4-{[(2,6-difluorophenyl)methyl]amino}-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-(furan-2-ylmethyl)-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[3-(pyridin-2-yl)propanoyl]piperidine-4-carboxamide
2-fluoro-5-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine-1-carbonyl]phenol
1-(7-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3-phenoxypropan-1-one
benzyl(cyclopropylmethyl)({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)amine
N-[(3R,4R)-3-hydroxy-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-4-yl]pyrazine-2-carboxamide
N-[3-(methylsulfanyl)propyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
(3R,4S)-N,N-dimethyl-4-(propan-2-yl)-1-(pyridine-3-sulfonyl)pyrrolidin-3-amine
2-[6-oxo-4-(1,2,3,4-tetrahydroisoquinolin-2-yl)-1,6-dihydropyridazin-1-yl]-N-[1-(thiophen-2-yl)ethyl]acetamide
2-(dimethylamino)-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-2-(3-methylphenyl)acetamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
7-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(methylsulfanyl)propan-1-one
N-ethyl-1-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1H-pyrrole-2-carboxamide