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1-(2,3-dihydro-1H-inden-2-yl)-4-{[(1,2-dimethyl-1H-imidazol-5-yl)methyl]amino}pyrrolidin-2-one
2-[4-(3-fluorophenyl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
3,5-dimethyl-7-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine
N-(3-{4-[(2,2-dimethyloxan-4-yl)amino]piperidin-1-yl}phenyl)-3-(trifluoromethyl)benzamide
6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N,N-dimethylpyrazine-2-carboxamide
4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-3-methyl-1-[(4-methylphenyl)methyl]piperazin-2-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-ethyl-N-methylacetamide
(1R,5R)-3-benzoyl-6-(1,3-thiazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[2-(butan-2-yl)phenoxy]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methylacetamide
1-(cyclohex-3-en-1-ylmethyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
5-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-ol
3-({1-azabicyclo[2.2.2]octan-3-yl}(pyridin-3-ylmethyl)amino)-N-cyclopropylpropanamide
2-[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-1-(piperazin-1-yl)ethan-1-one
3-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-7-methyl-1,2-dihydroquinolin-2-one
5-[(2-chlorophenyl)methyl]-5-[1-(3,3-dimethylbutanoyl)piperidin-4-yl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
3-[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propanoic acid
3-(1H-imidazol-4-yl)-2-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]formamido}propanoic acid
1-(1-cycloheptylpiperidin-3-yl)-3-(propan-2-yl)urea
1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)piperazine
1-(5-chloropyridin-2-yl)-4-(4-methanesulfonylbenzoyl)piperazine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(2-cyclohexylethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
5-{[4-(cyclohex-3-en-1-yl)-1H-1,2,3-triazol-1-yl]methyl}-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}oxy)benzamide
3-(hydroxymethyl)-1-(2,5,7-trimethylquinoline-4-carbonyl)piperidin-3-ol
1-[4-(3-cyclopentylpropyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecan-11-yl]-2-methylpropan-1-one
3-[(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)oxy]pyridine
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2,8-dimethylquinoline-4-carboxamide
N-phenyl-5-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-(4-{[4-(3-chloro-2-fluorobenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
1-methyl-N-[(3R,5S)-1-[(5-methylfuran-2-yl)methyl]-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
(1R,3S)-3-amino-N-[3-(4-chlorophenyl)propyl]cyclohexane-1-carboxamide
N-ethyl-2-{4-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]piperazin-1-yl}acetamide
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
1-{1-[3-(2-methoxybenzamido)phenyl]piperidin-4-yl}piperidine-3-carboxamide
3-{1-[(4-methylthiophen-2-yl)sulfonyl]piperidin-3-yl}benzoic acid
2-(cyclohex-1-en-1-yl)-1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)ethan-1-one
2,3-dimethyl-5-phenyl-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
2,5-dioxo-6-[3-(pyrrolidin-1-yl)butyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N,N-diethyl-3-{[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)sulfamoyl}benzamide
5-cyclobutyl-N-[2-(3,4-dimethoxyphenyl)ethyl]-1,3,4-oxadiazol-2-amine
5-{1-[(2-ethoxypyridin-3-yl)methyl]-1H-imidazol-2-yl}-2-(furan-2-yl)pyrimidine
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-dimethylacetamide
(1R,5R)-3-[4-(piperidin-1-ylmethyl)benzoyl]-3,9-diazabicyclo[3.3.2]decan-10-one
N-[1-(3-phenylpropyl)piperidin-3-yl]-2-(phenylsulfanyl)acetamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(2-methoxyphenyl)piperidine