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1-benzoyl-N-(4-fluorophenyl)piperidin-3-amine
6-chloro-N-{[2-(dimethylamino)pyridin-3-yl]methyl}quinolin-2-amine
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine
(2S)-N2-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidine-1,2-dicarboxamide
4-{2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}-N,N-dimethylpiperazine-1-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[(1-ethyl-1H-imidazol-2-yl)methyl]piperazine
1-(cyclopropylmethyl)-N-methyl-5-[(4-oxo-4H-chromen-3-yl)methyl]-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)propanamide
4-hydroxy-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
(2S,4S)-1-methyl-N-(pyridin-4-ylmethyl)-4-[(pyrrolidine-1-carbonyl)amino]pyrrolidine-2-carboxamide
8-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-(quinolin-5-ylmethyl)-1,2-oxazole-3-carboxamide
(1R,7S)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-oxo-3-(pentan-3-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-cyclopropyl-N-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[(6-ethoxypyridin-3-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
(5S,9aS,9bS)-5-[5-(methoxymethyl)furan-2-yl]-2-(2-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-methyl-N-(2-{7-[(5-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
2-{9-[(2-methoxyphenyl)carbamoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
(3aR,6aR)-2-cyclopropanecarbonyl-5-(pyridin-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(1H-pyrazol-1-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]benzamide
4-(1-benzofuran-2-sulfonyl)piperazine-2-carboxylic acid
[2-(2-fluorophenyl)ethyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanol
3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]propanamide
1-cyclopentyl-N3-ethyl-4-oxo-N5-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
2-[2-(1H-indol-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
4-(4-chlorophenyl)-N-methyl-N-(oxan-2-ylmethyl)butanamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(2-ethyl-1H-1,3-benzodiazol-1-yl)propan-1-one
5-methyl-6-(2-methylpiperidine-1-carbonyl)-N-(pyridin-2-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
4-[5-(methoxymethyl)furan-2-carbonyl]-1-(2-methoxyphenyl)-2,2-dimethylpiperazine
(2R,6R)-4-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-(dimethylamino)-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
[(3S,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(5-methylpyrazine-2-carbonyl)piperidin-3-yl]methanol
N-[2-(2-fluorophenyl)ethyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
(1S,6R)-3-methyl-9-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
ethyl 1-[(5-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]carbamoyl}-6-oxo-1,6-dihydropyridin-2-yl)methyl]piperidine-3-carboxylate
2-({[1-(5-chloro-2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-5-methyl-1,3,4-oxadiazole
1-[3-(3-methoxypiperidine-1-carbonyl)benzenesulfonyl]-4-methyl-1,2,3,6-tetrahydropyridine
(4aS,8aR)-6-(1H-imidazol-2-ylmethyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
2-acetyl-8-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidine
N-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carboxamide
1-(4-{5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
1-(furan-2-ylmethyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}piperidine-4-carboxamide
3-{5-[2-(1H-pyrrol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
1'-(2-fluoro-4-methylbenzoyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(2R)-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
3-(azepane-1-carbonyl)-1-ethyl-N-{[3-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-chloro-4-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-6-methoxyphenol
3-[(3-ethyl-1,2-oxazol-5-yl)methyl]-5-(piperidin-4-yl)-5-(pyridin-3-yl)imidazolidine-2,4-dione