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N-[2-(3-phenylpropoxy)phenyl]piperidine-4-carboxamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide
1-{2-[(1,4-dioxan-2-ylmethyl)(methyl)amino]pyrimidin-4-yl}piperidin-4-ol
N-tert-butyl-2-[6-(methoxymethyl)pyrimidin-4-yl]benzene-1-sulfonamide
3-{4-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
2-(2-{[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl}phenoxy)acetic acid
7-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-2-oxa-7-azaspiro[4.5]decane
(1R,7S)-3-(2-ethoxyethyl)-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-({[(3R,4R)-1-(2-amino-6-methylpyrimidin-4-yl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-4-(thiophen-2-yl)butanamide
N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(4-methyl-1,3-thiazol-5-yl)propanamide
4-[1-(1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]morpholine
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
2-(benzyloxy)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
1-(furan-2-ylmethyl)-N-methyl-N-(thian-4-yl)piperidine-3-carboxamide
1-{2-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-[1-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2H-1,3-benzodioxole-5-carboxamide
[(3R,4R)-1-(1H-indole-5-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
3-cyclopropyl-N-[(1R,3S)-3-[(2,3-dihydro-1H-inden-5-yl)carbamoyl]cyclopentyl]-1,2-oxazole-5-carboxamide
8-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(1-methyl-4-phenyl-1H-pyrazol-5-yl)-3-[2-(2-methylpropanesulfonyl)ethyl]urea
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
2-(1,3-benzoxazol-2-yl)-N-(thiolan-3-yl)acetamide
8-(morpholine-2-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-benzyl-8-(2-hydroxypyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(1-{3-[(3-chlorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidin-4-yl)(phenyl)methanol
N-benzyl-N-methyl{[(1S,2R)-2-(cycloheptylamino)cyclobutyl]amino}sulfonamide
2-methoxy-1-(4-{2-[2-(2-methoxyphenyl)ethyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)ethan-1-one
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,4-dimethyl-1,2,3-thiadiazole-5-carboxamide
methyl 6-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-5-cyano-2-methylpyridine-3-carboxylate
7-fluoro-3-({[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]amino}methyl)-1,2-dihydroquinolin-2-one
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
3-(benzyloxy)-1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
1-(cyclobutylmethyl)-3-({[(2-fluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
[1-(2-chlorobenzoyl)-3-[(2-methylphenyl)methyl]piperidin-3-yl]methanol
1-(4-methoxy-2-methylphenyl)-3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}urea
(1R,5R)-6-(cyclobutylmethyl)-3-(2-propyl-1,3-thiazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-{1-[2-(2,6-difluorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
N,N,3,6-tetramethyl-2-[2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-5-yl]quinoline-4-carboxamide
N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl 1-benzyl-5-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(3aS,6aS)-5-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(6-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-3-yl)ethan-1-one
(benzylsulfamoyl)(1,4-dioxan-2-ylmethyl)methylamine
N-({5-[(3-cyanophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
(5S,9aS,9bS)-5-(2-chlorophenyl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-{3-[(4-cyclohexylpiperazin-1-yl)methyl]-8-methylimidazo[1,2-a]pyridine-2-carbonyl}morpholine
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}quinoline
1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one