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4-(pyridin-2-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
(4aS,8aR)-6-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
2-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
N-cyclopentyl-2-cyclopropyl-4-methyl-N-[(5-methylthiophen-2-yl)methyl]pyrimidine-5-carboxamide
1-[1-(2-fluoro-6-methoxybenzoyl)piperidin-3-yl]-3-phenylpropan-1-one
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
1-{3-[(3,5-dimethyladamantan-1-yl)formamido]propyl}piperidine-4-carboxamide
N-(adamantan-2-ylmethyl)-6-{[butyl(methyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(naphthalen-1-ylmethyl)amine
methyl[(5-methylfuran-2-yl)methyl]{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}amine
4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperazine-1-sulfonamide
4-[4-(3,4-difluorophenyl)-5-methyl-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-methylpiperidine-4-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-(2H-1,3-benzodioxol-5-yloxy)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}acetamide
(2S)-N-[4-(3-fluorophenyl)phenyl]-1-[2-(morpholin-4-yl)ethyl]pyrrolidine-2-carboxamide
(3S)-3-acetamido-N-[2-(2-methoxyphenoxy)phenyl]pyrrolidine-1-carboxamide
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-5-methyl-6-(4-phenylpiperazine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
(4aR,7aS)-1-methyl-4-[(2-propoxynaphthalen-1-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({5-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
4-[(2-methylphenyl)methyl]-1-[(5-methylthiophen-2-yl)methyl]-1,4-diazepan-5-one
3-[(2-methylprop-2-en-1-yl)oxy]-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]benzamide
2-(1H-pyrazol-1-ylmethyl)-4-(1,3-thiazol-4-ylmethyl)-1,4-oxazepane
2-(4-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
6-chloro-3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-methylimidazo[1,2-a]pyridine
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-4-(1H-pyrazol-3-yl)benzamide
N,N-dimethyl-2-[methyl({[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl})amino]propanamide
1-[7-(3-chlorophenyl)-9-[(1-methylpiperidin-3-yl)methoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
(4aR,7aS)-1-benzyl-4-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[3-(furan-2-yl)-5-[1-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propyl]-1H-1,2,4-triazol-1-yl]acetic acid
N-{1-azabicyclo[2.2.2]octan-3-yl}-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
1-{1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]piperidin-3-yl}-3-phenylpropan-1-one
1'-[3-(1H-pyrazol-1-ylmethyl)benzoyl]spiro[indene-1,4'-piperidine]
1-(2,6-dimethylpyridin-3-yl)-3-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}urea
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]piperidin-4-ol
3-[(2-{2-[(propan-2-yl)carbamoyl]ethyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)methyl]-1,2,4-oxadiazole-5-carboxamide
2-{2-[5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazol-2-yl]phenoxy}acetamide
6-[(2,2-dimethyloxan-4-yl)amino]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(2-phenylethyl)acetamide
methyl 6-({[2-(morpholin-4-yl)pyridin-3-yl]methyl}amino)pyridine-3-carboxylate
3-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
(3S,4R)-4-(3-fluorophenyl)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]pyrrolidine-3-carboxylic acid
5-({[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
methyl (2S,4R)-1-[(2-hydroxyphenyl)methyl]-4-[3-(4-methylphenyl)propanamido]pyrrolidine-2-carboxylate
1-{3-[4-(2-amino-6-methylpyrimidin-4-yl)piperazine-1-carbonyl]piperidin-1-yl}ethan-1-one
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)cyclopropanecarboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]acetamide
N-methyl-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
7-(1,3-benzothiazol-2-yl)-9-hydroxy-N-(propan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
4-methyl-3-(3-{1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyridine