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6-methoxy-2-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]-1H-1,3-benzodiazole
2-hydroxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-(methylsulfanyl)butanamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
2-(2-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]formamido}ethyl)-4-methyl-1,3-thiazole-5-carboxylic acid
2-amino-N-[(3R,4S)-1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
1-{[2-(3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(1-methyl-1H-imidazol-2-yl)piperidine
[2-(1H-1,3-benzodiazol-2-yl)ethyl]({[2-(2,5-dimethoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl})amine
3-(azepane-1-carbonyl)-N-(furan-2-ylmethyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-({[(3R,4R)-1-(7-chloro-1-methyl-1H-indole-2-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[(7-{[2-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzenesulfonamide
2-(4-{[2-(5-methylfuran-2-yl)phenyl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
2-{3-methyl-5-[(2-methyl-1H-indol-3-yl)methyl]-1H-1,2,4-triazol-1-yl}acetic acid
1-{1-[(5-chlorofuran-2-yl)methyl]azetidin-3-yl}piperidine
7-(propan-2-yl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S,4R)-1-[5-(methoxymethyl)thiophene-2-carbonyl]-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
2-ethyl-N-[3-(1H-imidazol-1-yl)propyl]-6-methyl-1-[(5-methylfuran-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-[1-(4-methoxyphenyl)cyclopentyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[2-({[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]acetamide
4-acetyl-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-1,4-diazepane-1-carboxamide
2-benzyl-9-[2-(2-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1,3-benzothiazol-2-ylmethyl)-7-(2-methoxyacetamido)-1-methyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
1-{2-[2-(morpholin-4-ylmethyl)phenyl]pyrimidin-4-yl}piperidin-4-ol
N-[(1S,2R)-2-aminocyclobutyl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
2-{[4-(3-chlorophenyl)-5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-(2-{4-[(6-chloropyridin-3-yl)methyl]piperazin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-(4-methoxy-2-methylphenyl)-3-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]propanamide
3-(2-amino-1,3-thiazol-4-yl)-1-(6-hydroxy-1,4-oxazepan-4-yl)propan-1-one
dimethyl[(5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,3,4-oxadiazol-2-yl)methyl]amine
2-(benzyloxy)-1-[6-hydroxy-4-(1H-imidazol-2-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
N-ethyl-5-({3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)pyrimidin-2-amine
5,6-dimethyl-3-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-[2-(3-fluorophenyl)ethyl]-4-[4-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
5-methyl-N-[(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)methyl]-1,2-oxazole-3-carboxamide
5-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
N-[(2-methoxyphenyl)methyl]-2-[6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-2-yl]acetamide
1-(2,3-difluoro-6-methoxybenzoyl)-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
2-cyclopentyl-8-(5,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
methyl (2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxylate
3-(1H-imidazol-1-yl)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]butan-1-one
N-[3-(4-methylbenzamido)phenyl]-2,5-dihydro-1H-pyrrole-2-carboxamide
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](methyl)[(6-methylpyridin-2-yl)methyl]amine
1-(2-amino-6-methylpyrimidin-4-yl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)oxane-4-carboxamide
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-N-(pyridin-2-ylmethyl)cyclohexanamine
2-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-{[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-N,N-dimethylpyrimidin-2-amine
5-acetyl-N-(2-hydroxy-1-phenylethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2-oxoazepan-1-yl)acetamide
N-[(1S)-1-[1-tert-butyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]-2-(1H-imidazol-4-yl)ethyl]acetamide