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N-[2-(azepan-1-yl)ethyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-(propan-2-yl)acetamide
4-{[2-(1-cycloheptanecarbonylpiperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-6-azaspiro[2.5]octane-1-carboxamide
4-(3,4,5-trimethoxyphenyl)-1H-pyrrolo[2,3-b]pyridine
4-methyl-2-(piperidin-1-yl)-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]pyrimidine
4-fluoro-N-(2-{7-[(5-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
4-[2-(3,4,5-trimethoxyphenyl)acetyl]piperazine-2-carboxylic acid
2-[2,5-dioxo-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}acetamide
N-[2-(7-{[4-(methylsulfanyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]oxolane-2-carboxamide
N-(butan-2-yl)-3-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-4-ylmethyl)propanamide
3-(2-ethyl-1H-1,3-benzodiazol-1-yl)-1-[3-(phenylamino)piperidin-1-yl]propan-1-one
{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}(ethyl)({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amine
9-[2-(ethylamino)pyrimidine-5-carbonyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-1-(furan-3-ylmethyl)-6-[(3-hydroxyphenyl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
(4aR,7aS)-1-ethyl-4-[4-(1H-pyrazol-3-yl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2-methyl-6-propylpyrimidin-4-yl)-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperidin-4-amine
2-(pyridin-3-yl)-7-[2-(pyrrolidin-1-yl)butanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3S,4R)-N-(5-fluoro-2-methylphenyl)-3-hydroxy-4-(hydroxymethyl)piperidine-1-carboxamide
5-[2-(3,4-difluorophenyl)ethyl]-3-methyl-1-propyl-1H-1,2,4-triazole
1-(cyclohexylmethyl)-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-6-oxopiperidine-3-carboxamide
4-(6-ethyl-2-methylquinoline-4-carbonyl)-1-phenylpiperazin-2-one
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)furan-2-carboxamide
7-(3-chlorophenyl)-4-(2,2-dimethyloxane-4-carbonyl)-9-(pyridin-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2,5-dimethyl-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-[3-(5-methylfuran-2-yl)butyl]-4-(1H-pyrrole-2-carbonyl)piperazine
4-(1,3-benzothiazol-2-yl)-2-({[2-(1H-indol-3-yl)ethyl]amino}methyl)phenol
{1-[2-(methylsulfanyl)benzoyl]-4-(2-phenoxyethyl)piperidin-4-yl}methanol
N-(2-{7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-(4-fluorophenyl)acetamide
3-{[(4-chlorophenyl)methyl](3-hydroxypropyl)carbamoyl}benzoic acid
1-(5-chloropyridin-2-yl)-4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
2-(4-chlorophenyl)-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}morpholine
N-(1-ethyl-5-oxopyrrolidin-3-yl)-2-methoxy-2-phenylacetamide
4-[5-({3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}methyl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
3,5,7-trimethyl-2-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]-1H-indole
3-[4-(2,4-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2,4,6-trimethoxyphenyl)methyl]piperidine
1-methyl-3-[3-(4-{[3-(1H-pyrazol-1-yl)propyl]amino}piperidin-1-yl)phenyl]imidazolidin-2-one
(3aR,7aS)-2-(2-phenylmethanesulfonylbenzoyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-fluoro-N-(4-{4-[(1-phenylcyclopropyl)amino]piperidin-1-yl}phenyl)benzamide
2-[1-(6-aminopyridin-3-yl)-1H-pyrazol-4-yl]ethan-1-ol
2-(5-{6-chloroimidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
N,N,4-trimethyl-3-({[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
5-(2-fluorophenoxymethyl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
2-(4-hydroxy-3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[(3-fluorophenyl)methyl]-4-[3-(1H-imidazol-2-yl)benzoyl]piperazine
methyl 3-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[5-(5-chloro-2-methoxypyridin-4-yl)-1H-1,3-benzodiazol-2-yl]ethan-1-ol
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-hydroxybutan-1-one
N-[4-(4-{[(4-chlorophenyl)(pyridin-4-yl)methyl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
2-(morpholin-4-yl)-N-[2-(pyridin-2-yl)ethyl]-2-(pyridin-3-yl)acetamide
{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine