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2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}acetic acid
N-({4-hydroxy-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]azepan-4-yl}methyl)methanesulfonamide
1-[benzyl(methyl)amino]-3-(4-{[benzyl(methyl)amino]methyl}phenoxy)propan-2-ol
(5Z)-5-{2-[(4aR,8aR)-6-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridin-1-yl]-2-oxoethylidene}-1,3-thiazolidine-2,4-dione
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(pyridin-3-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-(1-benzofuran-5-yl)-4-hydroxy-4-(hydroxymethyl)azepane-1-carboxamide
1-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-hydroxypropan-1-one
4-methoxy-N-(2-{7-[(4-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
4-chloro-3-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1H-pyrazole-5-carboxamide
3-[3-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-5-methylpyridine
4-{4-[(2E)-2-methylbut-2-en-1-yl]piperazin-1-yl}-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
N,6-dimethyl-4-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1H-1,2,3-triazole-5-carboxamide
1-[(2-chloro-4-fluorophenyl)methyl]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-(1-phenoxyethyl)-5-(thiophen-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-{4-[1-(dimethylamino)ethyl]phenyl}-N-methylpyridine-4-carboxamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]propanamide
(1R,5R)-6-benzyl-3-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonane
2-methoxy-3-[3-(pyridin-4-yl)azetidine-1-carbonyl]pyridine
1-(cyclohex-3-ene-1-carbonyl)-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
3-[2-(2-ethylpiperidin-1-yl)-2-oxoethyl]-3-(3-fluorophenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
1-cyclobutanecarbonyl-4-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-1,4-diazepane
(3aS,7aR)-5-methyl-2-[2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
8-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
ethyl 4-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
3-(but-2-yn-1-yl)-5-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
(3S)-3-benzyl-4-[(2-fluoro-4,5-dimethoxyphenyl)methyl]piperazin-2-one
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-4-methylpyrimidin-2-amine
2-methoxy-N-[3-(4-{[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]benzamide
2-[methyl({4-methyl-5-[1-(piperidin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
1-benzyl-N3-[(3-chlorophenyl)methyl]-N5-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(1S,6R)-9-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
2-{[3-(2-hydroxyethyl)-4-(1-methylpiperidin-4-yl)piperazin-1-yl]methyl}phenol
3-({[1-(1,3-thiazol-4-ylmethyl)piperidin-4-yl]oxy}methyl)pyridine
7-methyl-3-{[1-(piperidin-1-yl)cyclopentyl]methyl}-3,4-dihydroquinazolin-4-one
2-{4-[(8-methoxyquinolin-2-yl)methyl]morpholin-3-yl}acetic acid
1-methyl-4-phenyl-3-[1-(thiophene-3-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{1-methyl-4-[(1-methyl-1H-indol-3-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[2-(dimethylsulfamoyl)ethyl]-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanamide
1-[(5-ethylpyridin-2-yl)methyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(4aR,7aS)-1-ethyl-4-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(pyridin-2-ylmethyl)-1,4-diazepane
3-[4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazin-1-yl]propanamide
2-ethyl-N-(naphthalen-2-yl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
ethyl 1-[(5-acetylthiophen-3-yl)methyl]-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylate
4-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1,2-dihydroquinolin-2-one
3-(3-methylbut-2-en-1-yl)-1-[2-(2H-1,2,3-triazol-2-yl)acetyl]piperidine-3-carboxylic acid
methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}){[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amine
4-benzyl-3-[1-(4-methoxypyrimidin-2-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[3-(ethoxycarbonyl)-3-[(2-methylphenyl)methyl]piperidine-1-carbonyl]pyridin-1-ium-1-olate