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3-{[3-(2-fluorophenoxymethyl)piperidin-1-yl]methyl}pyridine
1-ethyl-N-(7-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-5-methyl-1H-pyrazole-4-carboxamide
N,N-dimethyl-2-[(6-methyl-2-phenylpyrimidin-4-yl)amino]ethane-1-sulfonamide
2-{1-[(4-ethoxyphenyl)methyl]-4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[5-(ethylsulfanyl)-1,3,4-thiadiazol-2-yl]-2-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]acetamide
ethyl 3-[(2-fluorophenyl)methyl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine-3-carboxylate
N-{1-[1-(3-chloro-2-fluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
4-(4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}phenyl)-2-methylbutan-2-ol
4-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamido]-N-phenylpiperidine-1-carboxamide
N-cycloheptyl-3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
1-(dimethyl-1,2-oxazole-4-carbonyl)-3-propylpiperidine-3-carboxylic acid
(1s,4s)-4-[4-(2-phenylmorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexan-1-amine
3-amino-1-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propan-1-one
2-methoxy-5-(1-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-imidazol-2-yl)phenol
N-(6-methoxy-4-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)acetamide
(2S,4R)-N-cycloheptyl-1-[(2,4-dimethylphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
N5-[(3,4-difluorophenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(3R)-1-{[6-(3-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}pyrrolidin-3-ol
6-(3-ethoxyphenyl)pyridine-3-carbonitrile
1-[2-(2-methoxyphenoxy)ethyl]-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-3-[(dimethylamino)methyl]piperidin-3-ol
8-acetyl-2-(2-ethoxypyridine-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(2-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)pyridine
1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-3-methylbutan-1-ol
3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]-5-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-4-(1-methyl-1H-pyrazol-4-yl)pyrimidine
1-(2-oxo-2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethyl)azepan-2-one
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-methyl-3-(1-methyl-3-phenyl-1H-pyrazol-5-yl)urea
2-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-5,6-dimethylpyridine-3-carbonitrile
(3R,4R)-1-(5-methyl-1,2,4-oxadiazol-3-yl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-(2-chloro-6-fluorophenyl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}acetamide
(4-{5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenyl)methanol
3-(1-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidin-2-yl)pyridine
4-(1-benzyl-5-{[2-(trifluoromethyl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl)morpholine
4-{3-fluoro-8-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-(4-methylphenyl)piperazin-2-one
1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-N-methylpiperidine-2-carboxamide
(2-oxo-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)urea
8-[2-(3-chlorophenyl)acetyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(2-cyclohexylethyl)-3-hydroxy-3-[({[4-(hydroxymethyl)phenyl]methyl}amino)methyl]piperidin-2-one
2-{octahydropyrrolo[1,2-a]piperazin-2-yl}-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridine
4-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
3-phenyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-3-(pyridin-2-yl)propanamide
4-(2-methyl-1,3-thiazole-4-carbonyl)-2-{[5-(pyridin-2-yl)-1,2,4-oxadiazol-3-yl]methyl}morpholine
5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
2-[2-fluoro-6-(propan-2-yloxy)phenyl]-2-(4-methyl-1,4-diazepan-1-yl)acetic acid
4-{[1-(3-fluoropyridin-4-yl)piperidin-4-yl]methyl}morpholine
N-(4-{[4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenyl)acetamide
(1S,5R)-6-(1H-indol-5-ylmethyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(4aS,8aR)-1-(carboxymethyl)-6-(3-chloropyridin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid