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1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(4-methylbenzenesulfonyl)propan-1-one
(2S)-2-amino-3-(1H-imidazol-4-yl)-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]propanamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(6-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
7-(3,4-dimethoxyphenyl)-9-methoxy-4-{[4-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{2-[methyl({2-methylthieno[2,3-d]pyrimidin-4-yl})amino]ethyl}piperidin-2-one
1-(2-methylphenyl)-3-[1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]urea
1-{3-[(benzylamino)methyl]phenoxy}-3-(4-ethylpiperazin-1-yl)propan-2-ol
1-[2-(3-fluorophenyl)ethyl]-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-6-oxopiperidine-3-carboxamide
(3S,4S)-1-(1,4-dithiepan-6-yl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
3-[5-(quinoline-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-[1-(4-{[(5-phenyl-1,2-oxazol-3-yl)methyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]furan-3-carboxamide
2-methyl-4-{4-[4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]phenyl}butan-2-ol
4-[(3-fluoro-2-methylphenyl)methyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
(1R,2R,4R)-N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)acetamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[(6-hydroxypyrimidin-4-yl)methyl]acetamide
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}pyridine-2-carboxamide
1-[4-(morpholin-4-ylmethyl)phenyl]-3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
(3R,4R)-1-methyl-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
1-propyl-N-[2-(pyridin-2-yl)ethyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
methyl (1R,3S,3aR,6aS)-3-(6-methoxypyridin-3-yl)-5-methyl-1-(2-methylpropyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
6-methyl-5-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H-imidazol-2-yl}quinoline
2-methyl-N-{2-[3-(3-methylbutoxy)phenyl]ethyl}-1,3-thiazole-4-carboxamide
N-[2-(1,3-benzoxazol-2-yl)ethyl]-5-cyclobutyl-1,3,4-oxadiazol-2-amine
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-6-methyl-2-(piperidin-1-yl)pyrimidin-4-amine
(2-methoxyethyl)(propan-2-yl){[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
(4aR,7aS)-1-(pyridin-2-ylmethyl)-4-[2-(1H-1,2,4-triazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-methyl-8-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-(benzyloxy)-1-{4-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-1-yl}ethan-1-one
1-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-3-[(1,4-dimethylpiperazin-2-yl)methyl]urea
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
N-(2,4-dimethylphenyl)-N'-{2-[(3-methylpyridin-2-yl)amino]ethyl}propanediamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-methyl-2-oxopentanamide
2-{3-[2-(1-ethyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenyl}-5-methyl-1,3,4-thiadiazole
[(2S,6S)-4-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
methyl 2-[(1-benzyl-1H-imidazol-5-yl)methyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
(3R,4S)-4-propyl-1-(3-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-amine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]-2-methylpyrimidine-5-carboxamide
1-[2-(3-fluorophenyl)ethyl]-N-[3-(methylsulfanyl)propyl]-6-oxopiperidine-3-carboxamide
3-[1-cyclohexyl-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1λ6-thiolane-1,1-dione
(1R,5S)-8-(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)-3,8-diazabicyclo[3.2.1]octane
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2,5-dimethylfuran-3-carboxamide
1-{3-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
(4aS,8aS)-N-ethyl-4a-hydroxy-N-methyl-7-(pyrazin-2-yl)-decahydro-2,7-naphthyridine-2-sulfonamide
N-(1-{7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
1-[9-methoxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2,2-diphenylethan-1-one