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5-ethyl-1'-[5-(methoxymethyl)thiophene-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-methoxyethan-1-one
6-(2,5-dimethylfuran-3-yl)-N-[(2S)-2-hydroxypropyl]-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[(1R,2R)-1-[(pyrimidin-4-yl)amino]-2,3-dihydro-1H-inden-2-yl]acetamide
(1R,3S)-N3-ethyl-1,2,2-trimethyl-N1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]cyclopentane-1,3-dicarboxamide
methyl 1-ethyl-5-{[(4-methoxyphenyl)methyl]amino}-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(2,3-dimethylquinoxalin-6-yl)-3-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]urea
8-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-methoxy-N-({1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}methyl)benzene-1-sulfonamide
1-(pyridin-2-ylmethyl)-4-[4-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]pyrrolidin-2-one
2-cyclopropyl-N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[1-(4-{methyl[(4-phenyl-1,3-thiazol-2-yl)methyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]furan-3-carboxamide
4-{[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
4-(1,5-dimethyl-1H-indole-2-carbonyl)-3-(3-fluorophenyl)piperazin-2-one
5-{4-hydroxy-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
5-methyl-N-(2-methylpropyl)-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
[(4-{furo[3,2-c]pyridin-4-yloxy}phenyl)methyl]dimethylamine
4-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-phenyl-1H-imidazol-5-yl}phenol
5-(1-benzofuran-2-yl)-3-[4-(2-phenoxyethyl)piperazin-1-yl]-1,2,4-triazine
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-5-(hydroxymethyl)furan-2-carboxamide
N-cyclohexyl-5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-benzyl-2,3-dihydro-1H-isoindole-2-sulfonamide
N-[(3-fluoro-4-methylphenyl)methyl]-2-(1-methyl-3-oxopiperazin-2-yl)acetamide
3-[(3R,4S)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
2-oxo-1-phenyl-N-[3-(pyridin-4-yl)propyl]pyrrolidine-3-carboxamide
(3S,4S)-1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
4-(3,4-dimethylphenyl)-5-[3-(methylsulfanyl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
5-{[(2-chlorophenyl)methyl](2-methoxyethyl)carbamoyl}-1H-imidazole-4-carboxylic acid
methyl 2-[(butan-2-yl)sulfamoyl]-6-[(2,3,6-trifluorophenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[4-({[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)amino}methyl)thiophen-2-yl]ethan-1-one
N-(4-{[4-(4-fluorophenoxy)piperidin-1-yl]methyl}phenyl)acetamide
N-{2-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-2-oxoethyl}acetamide
2-(1-methyl-4-phenylpiperidine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}sulfonyl)-1,2,3,4-tetrahydroisoquinoline
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[(3-methylpyridin-4-yl)methyl]benzamide
N-{[2-(4-chlorophenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
6-[(E)-2-phenylethenyl]-2H-1,3-benzodioxole-5-carboxamide
2-{2,7-diazaspiro[4.5]decane-7-carbonyl}-N,4-dimethylaniline
N-[2-(benzyloxy)ethyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]benzamide
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-(3-methyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(4-benzylpiperazin-1-yl)-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-(2-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
(1S,5R)-3-benzyl-6-(5-methylpyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]-N-[2-(1H-pyrazol-4-yl)ethyl]piperidin-4-amine
1-{6-[3-(1-propyl-1H-pyrazol-3-yl)phenyl]pyridin-3-yl}ethan-1-one
2-ethyl-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one