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N-[(3S,4R)-1-[3-(difluoromethoxy)benzoyl]-4-propylpyrrolidin-3-yl]acetamide
3-{[2-(3-methoxypropyl)piperidin-1-yl]methyl}phenol
N-({7-[(3,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
(1S,4R)-2-({1-butyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}methyl)-2-azabicyclo[2.2.1]heptane
3-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(2,4,6-trimethylpyridin-3-yl)urea
5-{3-[(4-fluorophenyl)methoxy]azetidine-1-carbonyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole
4-[(2R)-2-amino-2-phenylacetamido]-N-ethylpiperidine-1-carboxamide
[(3R,4R)-1-(2-amino-6-methylpyrimidin-4-yl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-(5-chlorothiophen-2-yl)-1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-imidazole
N,N-dimethyl-3-({[5-(morpholine-4-carbonyl)pyridin-2-yl]amino}methyl)pyridin-2-amine
1-[(diethylcarbamoyl)methyl]-N-[(3-phenylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-[2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetyl]-4-phenoxypiperidine-4-carboxylic acid
N-[(2R,3R)-1'-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
N-[(1-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]acetamide
[(1-ethyl-1H-imidazol-2-yl)methyl][(5-fluoro-2,3-dimethyl-1H-indol-7-yl)methyl]amine
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2,5-dimethylfuran-3-carboxamide
1-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]-4-(3-fluorophenoxy)piperidine
2,5-dimethoxy-N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)benzamide
1-{6-hydroxy-4-[3-(1H-pyrazol-1-yl)propyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
N'-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)ethanediamide
4-{1-[(4-methoxynaphthalen-1-yl)methyl]azetidin-3-yl}pyridine
5-{4-[2-(2,4-difluorophenoxy)acetyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-(4-methyl-1,3-thiazol-5-yl)propanamide
4-[1-tert-butyl-5-(5-methyl-2H-1,2,3-triazol-4-yl)-1H-1,2,4-triazol-3-yl]benzamide
4-[(2-methoxyphenyl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(cyclopropylmethyl)-9-[2-(3-fluorophenoxy)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
9-[(2S)-2-(methylamino)propanoyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
[(3R,4R)-1-(3,4-dichlorobenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
2-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
3-(4-methylphenoxymethyl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
2-methyl-6-[5-(oxolan-3-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-1-yl]-1,3-benzothiazole
ethyl 5-(5-acetylthiophene-2-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N,N-diethyl-1-[4-(4-methylphenoxy)piperidine-4-carbonyl]pyrrolidin-3-amine
3-{5-[(2,6-difluorophenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyridine
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]propanamide
ethyl 4-{1-[2-(1-methylpiperidin-4-yl)acetyl]piperidin-3-yl}piperazine-1-carboxylate
1-[(3-methoxyphenyl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
1-[(4-chlorophenyl)methyl]-N-[2-(diethylamino)ethyl]-6-oxopiperidine-3-carboxamide
ethyl 3-[(2-fluorophenyl)methyl]-1-[3-(2-oxopyrrolidin-1-yl)propanoyl]piperidine-3-carboxylate
2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(thiophen-2-yl)ethyl]acetamide
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
methyl (2S)-2-{[5-(2-fluorophenyl)-1,2,4-triazin-3-yl]amino}-3-methylbutanoate
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-(N-methylmethanesulfonamido)ethyl]propanamide
N4-methyl-N4-[(2-methylpyridin-4-yl)methyl]-6-(propan-2-yl)pyrimidine-2,4-diamine
2-cyclopentanecarbonyl-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
3-[1-(2-hydroxyacetyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
3-{4-[4-(methylamino)pyrimidin-2-yl]piperazin-1-yl}pyrazine-2-carbonitrile
4-{[5-(1-cyclopropanecarbonylpiperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}morpholine
1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane