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1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-methyl-N-propylpiperidine-3-carboxamide
2-methoxy-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]pyridine-3-carboxamide
2-[(2-fluorophenyl)methyl]-N-(2-phenoxyethyl)-1,3-benzoxazole-6-carboxamide
N-({1-[(3-hydroxyphenyl)methyl]pyrrolidin-3-yl}methyl)-2-(piperidin-1-yl)acetamide
N-(6-methoxyquinolin-8-yl)-3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine-1-carboxamide
2-methyl-6-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2,3-dihydropyridazin-3-one
N-[4-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}piperidin-1-yl)phenyl]-2-fluorobenzamide
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-(pyrazine-2-carbonyl)piperidin-4-ol
N-[(3S)-1-benzylpyrrolidin-3-yl]-5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-(furan-3-ylmethyl)piperidine
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-1-methyl-1H-pyrazole-5-carboxamide
9-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}pyridine-3-carboxamide
1-(2-benzylphenyl)-3-[(1,3-dimethylpyrrolidin-3-yl)methyl]-3-methylurea
1-[2-({2-methylpyrido[2,3-d]pyrimidin-4-yl}amino)ethyl]imidazolidin-2-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(5-ethylpyridin-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
ethyl 4-({7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}amino)benzoate
1-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]-3-methylimidazolidin-2-one
N-[(3R,4R)-3-hydroxy-1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl]pyridine-2-carboxamide
3-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-N-(3-chloro-4-fluorophenyl)propanamide
1-(4-chlorophenyl)-N-{[1-(pyrimidin-5-ylmethyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(isoquinolin-1-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
2-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-2-azaspiro[4.4]nonane
2,2-dimethyl-1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]propan-1-one
N-(4-carbamoyl-3-chlorophenyl)-3-(hydroxymethyl)piperidine-1-carboxamide
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-[2-(3-chlorophenyl)ethyl]-2-{[(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]amino}acetamide
4-(1-ethyl-1H-pyrazole-5-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 7-oxo-3-(1,3-thiazole-5-carbonyl)-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
9-methoxy-4-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3R,4R)-4-hydroxypyrrolidin-3-yl]-5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[(5-methylpyrazin-2-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
1-acetyl-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)piperidine-4-carboxamide
6-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrazolo[1,5-a]pyrimidine-3-carbonitrile
3-{[1-(3-fluorophenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
methyl 2-{2-[4-(3-cyanopyrazin-2-yl)piperazin-1-yl]acetamido}-4-methyl-1,3-thiazole-5-carboxylate
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
3-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetamido]-4-chloro-N,N-diethylbenzamide
1-(4-chlorophenyl)-5-methyl-4-(quinoline-3-carbonyl)piperazin-2-one
(2S,4S)-4-amino-N,N-diethyl-1-[(5-methylnaphthalen-1-yl)methyl]pyrrolidine-2-carboxamide
2-(4-methoxyphenoxymethyl)-N-[(3-methylphenyl)methyl]-1,3-oxazole-4-carboxamide
N-({1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}methyl)acetamide
[(2-chlorophenyl)methyl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
S-(2-benzoyl-1,2,3,4-tetrahydroisoquinolin-7-yl)-3-hydroxybutane-1-sulfonamido
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
(2S,4R)-1-[(3-chlorophenyl)methyl]-N,N-diethyl-4-{[(4-phenylphenyl)methyl]amino}pyrrolidine-2-carboxamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3R,4S)-1-(3-fluoro-4-methylbenzenesulfonyl)-4-propylpyrrolidin-3-amine
2-(1,4-dimethylpiperazin-2-yl)-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)acetamide