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3-methyl-8-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1R,5R)-6-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-[2-(4-cyclopentylpiperazin-1-yl)-2-oxoethyl]-4-[(3,5-dimethoxyphenyl)methyl]piperazin-2-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(2-oxopiperidin-1-yl)propanamide
2-cyclopropyl-1-[3-(2-phenylethyl)piperidin-1-yl]ethan-1-one
(1R,5S)-6-[3-(1,4-oxazepane-4-sulfonyl)benzoyl]-6-azabicyclo[3.2.1]octane
2-(adamantan-1-yl)-5-(morpholine-4-carbonyl)pyrimidin-4-ol
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-methoxypyridine-3-carboxamide
2-(3-fluorophenyl)-5-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-1,3,4-oxadiazole
5-[5-(piperidine-1-carbonyl)furan-2-yl]pyrimidine
1-(difluoromethyl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
(2S)-2-{[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-3-methylbutanamide
methyl 2-(1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
N-(2,3-dihydroxypropyl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
3-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-4-[(2-methylphenyl)methyl]piperazin-2-one
2-(2,6-dimethylpyridin-4-yl)-6-methoxy-N,N-bis(propan-2-yl)benzamide
1-{2-[5-(2-fluoro-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyrrolidin-2-one
1-methyl-N-[2-(N-methylmethanesulfonamido)ethyl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
3,5-dimethyl-4-[1-(thiophen-3-ylmethyl)pyrrolidin-2-yl]-1,2-oxazole
(3R,4R)-1-(6-ethylpyrimidin-4-yl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}acetamide
methyl (2S)-2-({4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]phenyl}formamido)-2-phenylacetate
2-(1-benzofuran-2-yl)-N-(propan-2-yl)pyrimidin-4-amine
N-{[7-fluoro-5-(quinolin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
(3R,4S)-4-(4-methoxyphenyl)-1-[3-(5-methylfuran-2-yl)benzoyl]pyrrolidin-3-amine
(3S,4S)-1-[(5-cyclopentylthiophen-2-yl)methyl]-4-methylpiperidine-3,4-diol
(3aR,6aS)-N-[3-fluoro-5-(trifluoromethyl)phenyl]-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
2-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-4,6-dimethylpyridine-3-carbonitrile
4-{[2-(dimethylamino)ethyl]amino}-5-methyl-N-{[4-(trifluoromethoxy)phenyl]methyl}thieno[2,3-d]pyrimidine-6-carboxamide
3-({4-[3-(2,2-dimethylpyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-({4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-6-methylpyridine
1-(dimethyl-1,3-oxazole-4-carbonyl)-3-(4-fluorophenoxymethyl)piperidine
4-{2-[2-(2,5-dichlorophenyl)-1H-imidazol-1-yl]propyl}morpholine
(3aR,6aR)-2-(2-methoxyacetyl)-N-[(3-methyl-1H-pyrazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(1R,3S)-3-{[2-(benzylsulfanyl)ethyl]carbamoyl}cyclopentane-1-carboxylic acid
8-[(2-methyl-1,3-benzothiazol-6-yl)sulfonyl]-1-oxa-8-azaspiro[4.5]decane
N-{2-[(2-ethylphenyl)carbamoyl]phenyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-(4-{[2-(furan-2-yl)phenyl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
(1S,6R)-N-(4-methyl-2-oxo-1,2-dihydroquinolin-7-yl)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
ethyl 5-{[(2R,3R)-2-ethoxy-3-propanamido-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]carbonyl}-2,4-dimethyl-1H-pyrrole-3-carboxylate
2-(4-methyl-1H-pyrazol-1-yl)-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-one
N-(adamantan-2-ylmethyl)-2-oxo-6-(piperidin-1-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-(4-fluorophenyl)-4-(2-methoxypyridine-3-carbonyl)-1,4-diazepane
4-[(5-ethyl-4-phenyl-1H-imidazol-1-yl)methyl]-3,5-dimethyl-1,2-oxazole
1-(2-oxo-2-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)pyrrolidin-2-one
4-(4-{[4-(4-chlorophenyl)phenyl]methyl}piperazin-1-yl)butan-1-ol
(3R,4S)-4-cyclopropyl-1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-3-amine
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(isoquinolin-5-ylmethyl)-N-methylpropanamide
(3S)-3-({[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)azepan-2-one