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3-(2-amino-1,3-thiazol-4-yl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)propanamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
2-[({[(2R,3R,5S)-2-(2-fluorophenyl)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]methyl}amino)methyl]-4-methoxyphenol
(4aR,7aS)-6,6-dioxo-N-[4-(1H-pyrazol-5-yl)phenyl]-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(2R)-2-cyclohexyl-N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-hydroxyacetamide
4-[5-(2-fluorobenzoyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
2-{4-[3-(5-methylfuran-2-yl)butyl]piperazin-1-yl}pyridine-3-carboxamide
1-{4-[({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]thiophen-2-yl}ethan-1-one
{4-[2-(2-phenylethyl)piperidine-1-carbonyl]phenyl}methanol
2-cyclopropyl-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2-{[4-(1,3-diphenyl-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]methyl}morpholine
methyl 5-[4-(4-methylphenoxy)piperidin-1-yl]-5-oxopentanoate
4-(2-methoxyphenoxy)-1-(oxane-4-carbonyl)piperidine
3-({[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]carbamoyl}amino)-N,2-dimethylbenzamide
N-(1-ethyl-1H-1,2,4-triazol-5-yl)-3-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}benzamide
(2R)-N-[2-(4-fluorophenyl)ethyl]-N-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
N-(3-{[butyl(furan-2-ylmethyl)carbamoyl]methoxy}phenyl)propanamide
2-[4-(2-methoxyethyl)piperazin-1-yl]-2-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}acetic acid
(2R)-1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-hydroxy-2-phenylethan-1-one
1-methyl-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]piperidine-3-carboxamide
{[5-(3-fluoropyridin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
2,6-dimethoxy-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]pyridine-3-carboxamide
5-[(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)methyl]quinoline
1-[2-(4-methoxy-3-methylphenyl)pyrimidin-4-yl]piperidin-3-ol
4-(1H-pyrazol-1-yl)-1-[3-(pyridin-3-yl)propanoyl]piperidine-4-carboxylic acid
N-[2-(1H-imidazol-4-yl)ethyl]-5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carboxamide
2-[1-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
2-(4-{[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
7-(6-ethyl-2-methylquinoline-4-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-(cyclohex-1-en-1-ylmethyl)-7-(1H-imidazol-4-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[2-(propan-2-yl)pyrimidine-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4R)-4-(4-{[1-(2,5-dimethylfuran-3-yl)-N-methylformamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
N-[2-(pyrazin-2-yl)ethyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
3-(1-methyl-1H-pyrrol-2-yl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-pyrazole-5-carboxamide
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-1,4-dithiepan-6-amine
3-[4-(1-carbamoylpiperidine-3-carbonyl)piperazin-1-yl]benzoic acid
4-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
6-[(3-methoxyphenyl)methoxy]-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
methyl 1-{2-hydroxy-3-[4-({[2-(1H-imidazol-1-yl)ethyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
(3R,4R)-1-({4-[methyl(phenyl)amino]phenyl}methyl)-4-(4-methylpiperazin-1-yl)piperidin-3-ol
5-(3,3-diphenylpiperidine-1-carbonyl)pyridin-2-amine
1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
4-ethyl-1-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[(4-methylphenyl)methyl]-5-{3-oxo-3-[4-(thiophene-2-carbonyl)piperazin-1-yl]propyl}pyrrolidin-2-one
1-(4-{3-[(dimethylamino)methyl]-3-hydroxypiperidine-1-carbonyl}phenyl)pyrrolidin-2-one
2-[N-(4-methylphenyl)methanesulfonamido]-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}acetamide
(1R,3S)-3-methoxy-7-[4-(4-methylpiperazin-1-yl)benzoyl]-7-azaspiro[3.5]nonan-1-ol
4-methyl-6-(4-{methyl[(3-phenyl-1H-pyrazol-5-yl)methyl]amino}piperidin-1-yl)pyrimidin-2-amine
2-{2-[5-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyridine
5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]pyridine-2,4-diol