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4-({4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}methyl)quinoline
4-[3-(1-methoxyethyl)phenyl]-6-methylpyrimidin-2-amine
N-[3-(4-fluorophenyl)phenyl]-1-(6-methylpyridine-3-carbonyl)piperidine-3-carboxamide
3-{[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrazole
6-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
3-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
(1S,5R)-6-(cyclobutylmethyl)-3-[(4-methoxypyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(4aS,8aR)-6-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
(1S,5R)-6-propyl-3-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aS,8aR)-6-[2-(4-fluorophenoxy)ethyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
ethyl 1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylate
2-benzoyl-N-(5-methyl-1,3,4-thiadiazol-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
4-{[2-(1-cyclopentanecarbonylpiperidin-4-yl)-1H-imidazol-1-yl]methyl}pyridine
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-1,5-dimethyl-1H-pyrrole-2-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)-2-(1H-pyrazol-1-yl)acetamide
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazole
3-[(3R,4S)-1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-{2-[4-(trifluoromethyl)phenyl]ethyl}piperidine-3-carboxamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N2,N2,N4-trimethyl-N4-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-{4-[(2-methoxyethyl)carbamoyl]-2-methylphenyl}-2-methylpyrrolidine-1-carboxamide
methyl 2-({2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}amino)acetate
methyl[(3-methylthiophen-2-yl)methyl]{[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
4-fluoro-1-[7-(1,2-oxazole-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidine
2-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
N-[1-(7-{[3-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-2-methylpropyl]-2-methoxyacetamide
1-[(2,3-dimethoxyphenyl)methyl]-3-{[(furan-3-ylmethyl)(methyl)amino]methyl}-3-hydroxypiperidin-2-one
2-{1-[(2-methylphenyl)methyl]-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
N-{[5-methyl-2-(4-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}-1,3-thiazole-4-carboxamide
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
N-[(6-methylpyridin-2-yl)methyl]-1-[4-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidine
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-3-methylpiperidine
2-{[(3-methyl-1,2-oxazol-5-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[(2,3-dimethoxyphenyl)methyl]-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
1-{4-[(6-chloro-4-{[(2,3-dimethoxyphenyl)methyl]amino}quinazolin-2-yl)methyl]piperazin-1-yl}ethan-1-one
5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
7-[(4-fluorophenyl)methyl]-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-{[4-(dimethylamino)oxan-4-yl]methyl}-3-[2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
6-butyl-2-[4-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
N-[4-(4-{[2-(1H-indol-3-yl)ethyl]amino}piperidin-1-yl)phenyl]-2H-1,3-benzodioxole-5-carboxamide
4-({4-methyl-5-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
5-(dimethylamino)-2-(2-oxo-2-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)-2,3-dihydropyridazin-3-one
4-{2-[1-(5-ethyl-1,3-oxazole-4-carbonyl)piperidin-2-yl]ethyl}phenol
9-(4-chloro-3-methylbenzoyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
2-[2-(2,4-dimethyl-3-oxopiperazin-1-yl)-2-oxoethyl]-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
N-[(3,4-difluorophenyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)azepan-4-amine
N-[1-(1-benzylpiperidin-4-yl)-2-(2-fluorophenyl)ethyl]-N,2-dimethylfuran-3-carboxamide
1-[4-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)thiophen-2-yl]ethan-1-one