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3-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-methyl-1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
5-ethyl-5-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
N-[(4-chlorophenyl)methyl]-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
2-{[(3R,5S)-1-(cyclohexylmethyl)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]pyrrolidin-3-yl]sulfanyl}-1H-1,3-benzodiazole
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-5-(oxolan-2-yl)thiophene-2-carboxamide
N-[2-(2-fluorophenyl)-1-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-4-yl]ethyl]-N-methyl-3-(methylsulfanyl)propanamide
5-propyl-3-[2-(pyridin-2-yl)ethyl]-5-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[2-(4-methoxyphenyl)ethyl]-2-(methylamino)-N-(pyridin-2-ylmethyl)pyridine-3-carboxamide
ethyl 4-[1-(1-methylcyclopropanecarbonyl)piperidin-3-yl]piperazine-1-carboxylate
3-(4-{4-[(3,3-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}piperidine-1-carbonyl)-N-methylpyridin-2-amine
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-ol
1-cyclohexyl-4-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperazine
2-(3-fluorophenyl)-1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]piperidine
2-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}-5-methoxyphenol
5-(2-{5-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-4-phenyl-1H-imidazol-1-yl}ethyl)-1H-1,2,3,4-tetrazole
3-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-9-hydroxy-4H-pyrido[1,2-a]pyrimidin-4-one
(4aR,7aS)-1-(2-methoxyacetyl)-4-[2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]-4-(trifluoromethyl)pyrimidine
N,N-diethyl-1-[4-(methylamino)pyrimidin-2-yl]piperidine-3-carboxamide
3-{5-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
1-[1-(5-chloro-2-fluorobenzoyl)piperidin-3-yl]-2-phenylethan-1-one
4-fluoro-N-{3-oxo-3-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propyl}benzamide
3-{[7-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine
N,2,3,6-tetramethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]quinoline-4-carboxamide
N1-(5-methylpyridin-3-yl)-4-(piperidin-1-yl)piperidine-1,4-dicarboxamide
5-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]-2-butyl-1,3-benzoxazole
2-amino-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]-5H-indeno[1,2-b]pyridine-3-carbonitrile
[2-(1H-imidazol-1-yl)ethyl]({[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl})methylamine
(3S,4R)-4-phenyl-1-(3-phenyl-1,2-oxazole-5-carbonyl)pyrrolidine-3-carboxylic acid
N-cyclohexyl-3-{[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]amino}propanamide
5-(butan-2-yl)-1-(2-hydroxyethyl)-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(2S,4S)-4-amino-N-methyl-1-{2-[(pyridin-2-ylmethyl)amino]benzoyl}pyrrolidine-2-carboxamide
5-chloro-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
5-ethyl-3-(2-methylprop-2-en-1-yl)-5-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
4-chloro-3-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]-1-methyl-1H-indazole
2-(2H-1,3-benzodioxol-5-yloxy)-1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]ethan-1-one
4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}thiomorpholine
4-({4-[(benzyloxy)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1-methyl-1H-pyrazole
2-(methylsulfanyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}benzamide
N,N-dimethyl-1-(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carbonyl)pyrrolidin-3-amine
(1R,5R)-3-methanesulfonyl-6-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[(5-fluoro-2-methylphenyl)methyl]amino}piperidin-1-yl)benzamide
4-methyl-2-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
2-[3-oxo-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-4-carboxamide
N,N-diethyl-2-{4-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}acetamide
4-[4-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperazin-1-yl]quinazoline
1-(2-fluorophenyl)-4-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperazine
5-[1-(2-cyclopentylacetyl)piperidin-4-yl]-3-(cyclopropylmethyl)-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione