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3-(2-{3-[(2-methylphenyl)methoxy]azetidin-1-yl}-2-oxoethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-cycloheptyl-N-methyl-N-(1,2-oxazol-5-ylmethyl)-6-oxopiperidine-3-carboxamide
[(3R,4R)-1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-1-ethylpyrrolidin-2-one
N-(propan-2-yl)-2-[3-(pyridin-3-yl)azetidin-1-yl]pyridine-4-carboxamide
2-[3-(naphthalene-2-carbonyl)piperidine-1-carbonyl]pyrazine
5-(1-{2-methyl-3-[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]propyl}-1H-1,2,3-triazol-4-yl)pyrimidine
1-[4-(1H-pyrazol-3-yl)benzoyl]-4-(4H-1,2,4-triazol-3-yl)piperidine
N-[(3-hydroxy-4-methoxyphenyl)methyl]-N-methyl-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-(2-fluorophenyl)-N-methyl-1H-pyrazole-4-carboxamide
3-(2-methylpropyl)-N-[1-(thiophen-2-yl)propan-2-yl]-1,2-oxazole-5-carboxamide
N-[2-(4-methoxyphenyl)propan-2-yl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylpyridine-2-carboxamide
4-{1-[(2-ethylphenyl)methyl]piperidin-4-yl}pyrimidin-2-amine
N-[(3R,4S)-4-cyclopropyl-1-(2-hydroxyethyl)pyrrolidin-3-yl]-3-(4-fluorophenyl)propanamide
1-[(2-fluorophenyl)methyl]-N-methyl-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-3-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{5-[(dimethylamino)methyl]furan-2-carbonyl}-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
ethyl 4-({6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1H-pyrazole-3-carboxylate
3-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]-5-chloro-4,6-dimethyl-1,2-dihydropyridin-2-one
2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-[1-(thiophen-3-yl)propan-2-yl]acetamide
1-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-4-phenylbutan-1-one
2-methyl-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-1-benzofuran-5-carboxamide
1-({1-[6-(azocan-1-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
5-acetyl-N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]thiophene-3-carboxamide
methyl[(5-phenyl-1,2-oxazol-3-yl)methyl]{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amine
3-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-1-(2-methoxyethyl)pyrrolidine
2-(4-fluorophenoxymethyl)-N-[2-(oxan-2-yl)ethyl]-1,3-oxazole-4-carboxamide
ethyl({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl})[(1-methyl-1H-pyrazol-4-yl)methyl]amine
[(3R,5S)-1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
1-{4-[(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)methyl]phenyl}ethan-1-one
5-hydroxy-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrazine-2-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-4-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
4-benzyl-3-ethyl-1-(1H-indole-6-carbonyl)-1,4-diazepan-5-one
1-(4-{[4-(benzyloxy)piperidin-1-yl]methyl}phenyl)imidazolidin-2-one
N-(oxolan-3-yl)-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
(3R,4R)-1-[2-(dimethylamino)benzoyl]-4-ethylpiperidine-3,4-diol
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
[(2S,6S)-4-[(2-fluorophenyl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
2-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-phenylpropan-1-one
1-[(5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-2,4-dimethylphenyl)methyl]-4-methylpiperazine
N-(propan-2-yl)-5-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
3-(2-methylphenyl)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]pyrrolidin-3-ol
4-ethyl-1-methyl-3-{1-[(4-methylthiophen-2-yl)sulfonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1,3-thiazole-4-carboxamide
N-{3-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}acetamide
1-[3-(2-oxopyrrolidin-1-yl)propyl]-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidin-2-one
3-fluoro-N-({7-[(2,4,5-trimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
2-{[(4aS,8aR)-2-oxo-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-6-yl]methyl}benzonitrile