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butyl 2-benzoyl-4-oxo-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxylate
N-(1,4-dithiepan-6-yl)-1-[(2-fluorophenyl)methyl]piperidin-3-amine
ethyl 4-[(4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperazine-1-carboxylate
N-(6-phenoxypyridin-3-yl)-1-(pyridin-4-ylmethyl)piperidine-4-carboxamide
6-[4-(aminomethyl)phenyl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
2-(2-{[propyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)acetamide
[(2-ethoxyphenyl)methyl](methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
[1-(1-benzofuran-2-ylmethyl)-3-(2-phenylethyl)piperidin-3-yl]methanol
methyl 1-{2-[(2-ethylpiperidin-1-yl)methyl]-6,7-dimethoxyquinazolin-4-yl}piperidine-4-carboxylate
4-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2-(3-phenylpropyl)morpholine
{[2-(2-methylphenoxy)pyridin-3-yl]methyl}[(2-methylpyrimidin-5-yl)methyl]amine
6-[1-(4-chlorophenyl)cyclobutanecarbonyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxylic acid
4-fluoro-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-[1-(4-fluorophenyl)-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-2-(methylamino)acetamide
N-ethyl-3-({[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}sulfamoyl)-N-methylbenzamide
(1S,5R)-6-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
(3S,4R)-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]-4-phenylpyrrolidine-3-carboxylic acid
N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}oxane-4-carboxamide
N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1-benzothiophene-2-carboxamide
N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-(3-fluorophenyl)-1,2,4-triazin-3-amine
5-methyl-1-propyl-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
1-{2-[(dimethylamino)methyl]benzoyl}-3-(2-methoxyethyl)piperidine-3-carboxylic acid
1-(2-phenoxypropanoyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-9H-purin-6-amine
N-[(4-cyanophenyl)methyl]-2-(2-oxopiperidin-1-yl)acetamide
3-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-1H-pyrazol-5-amine
ethyl 1-benzyl-5-[2-(thiophen-2-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
5-methyl-N-[1-(pyrazin-2-yl)piperidin-4-yl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
N-(2,4-dimethoxyphenyl)-3-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}propanamide
ethyl 3-(2-methoxyethyl)-1-{[3-(methylsulfanyl)phenyl]methyl}piperidine-3-carboxylate
2-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}-6-methoxyphenol
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(3-methylthiophene-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(4aS,7aR)-1-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)methyl]-1-(propan-2-yl)-1H-pyrazole
4-[3-(propan-2-yl)-1H-pyrazol-1-yl]-1-(pyrrolidine-1-carbonyl)piperidine-4-carboxylic acid
N-(2-hydroxy-3-methoxypropyl)-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
8-(2-hydroxyacetyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
4-[1-cyclohexyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-1-cyclopentylpyrrolidin-2-one
2-{2-methoxy-4-[(3-oxo-4-phenylpiperazin-1-yl)methyl]phenoxy}acetamide
1-{2-methyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-4-phenylbutane-1,2-dione
4-[5-(propan-2-yl)pyrimidin-4-yl]-2-(trifluoromethyl)morpholine
1-[3-(difluoromethoxy)phenyl]-3-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}urea
methyl (2S,4S)-1-[(2-fluorophenyl)methyl]-4-[4-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
3-{4-[3-methoxy-5-(trifluoromethyl)phenyl]-3,5-dimethyl-1H-pyrazol-1-yl}propanamide
6-methyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}pyridine-2-carboxamide
1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)methanesulfonamide
3-chloro-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
1-[6-(dimethylamino)pyrimidin-4-yl]-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylic acid