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5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}furan-2-carboxamide
N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-[3-(5-chloro-1H-1,3-benzodiazol-2-yl)propyl]-3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)urea
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
benzyl(cyclopropylmethyl){[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}amine
1-[4-(pyridin-4-yl)piperidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}({[1-(piperidin-1-yl)cyclohexyl]methyl})amine
1-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
5-(methoxymethyl)-N-({3-methyl-7-[2-(piperidin-1-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
N-[(3S,4R)-1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(4-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]ethan-1-one
[4-({1-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyridin-2-amine
5-(2-chlorophenyl)-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]furan-2-carboxamide
N-methyl-3-(2-oxoazepan-1-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
(1-{3-[2-(pyridin-3-yl)-1H-imidazol-1-yl]propyl}piperidin-2-yl)methanol
3-phenoxy-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
methyl 4-({5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazol-3-yl}formamido)butanoate
3-({[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}amino)-N-(2-ethylphenyl)propanamide
1-ethyl-4-{2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-3-methylpiperazin-2-one
(4aS,8aR)-6-(4-methylpyrimidin-2-yl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
2-[1-(1-cyclobutanecarbonylpiperidine-4-carbonyl)piperidin-2-yl]pyridine
2-(dimethylamino)-8-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
(2S,4R)-N,N-diethyl-4-(2-methoxy-4-methylbenzamido)-1-methylpyrrolidine-2-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[2-(4-hydroxyphenyl)ethyl]-5-methoxybenzamide
1-{2-methoxy-4-[(4-phenylpiperazin-1-yl)methyl]phenoxy}-3-(morpholin-4-yl)propan-2-ol
1-[2-methyl-7-(3-methylfuran-2-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]pyrrolidine
1-(7-{[2-(hydroxymethyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(3,4,5-trimethoxyphenyl)ethan-1-one
2-{2-[4-(2-amino-1,3-benzothiazole-5-carbonyl)piperazin-1-yl]ethoxy}ethan-1-ol
2-amino-4-(3,4-dihydroxyphenyl)-6-(2-fluoro-4-methoxyphenyl)pyridine-3-carbonitrile
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2-(2-oxo-1,2,3,4-tetrahydroquinolin-1-yl)acetamide
2-amino-6-cyclobutyl-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)pyridine-3-carbonitrile
1-(6-carbamoylpyrazin-2-yl)-4-(4-methylphenoxy)piperidine-4-carboxylic acid
N-[3-(3-methoxyphenyl)phenyl]-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidine-4-carboxamide
methyl 6-{[benzyl(3-hydroxy-2-methylpropyl)amino]methyl}pyridine-2-carboxylate
4-(1-butyl-1H-imidazol-2-yl)-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidine
2-amino-4-propyl-6-(pyridin-3-ylmethyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1,2-dimethyl-3-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}-1H-indol-5-ol
methyl 4-{5-chloro-2-[(oxan-4-ylformamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}benzoate
N-({1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
5-[(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-2-methoxyphenol
[(dimethyl-1,2-oxazol-4-yl)methyl][1-(dimethyl-1,3-thiazol-4-yl)ethyl]methylamine
5-(4-cyclohexylphenyl)-N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-1,2,4-triazin-3-amine
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-(pyridine-2-carbonyl)piperidin-4-amine
1-[6-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)pyridin-2-yl]ethan-1-ol
1-cyclopropyl-4-[5-(2,4-dimethylphenyl)-4-methyl-1H-imidazol-2-yl]pyrrolidin-2-one
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2-(1H-pyrazol-1-yl)benzamide
methyl (2S)-1-{4-[4-(furan-3-amido)-1H-pyrazol-1-yl]benzoyl}pyrrolidine-2-carboxylate
N-(2-methoxy-5-methylphenyl)-2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide