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1-cyclobutanecarbonyl-4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1,4-diazepane
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(2-methoxyphenyl)-2-methylpiperazine
N-[(5-fluoro-2-oxo-2,3-dihydro-1H-indol-3-yl)methyl]-2-(1H-pyrazol-1-yl)acetamide
1-[1'-(1-ethyl-1H-pyrazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N-[2-(diethylamino)ethyl]-N-ethyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carboxamide
3-(4-{[3-(2-phenylpyridin-4-yl)pyrrolidin-1-yl]methyl}phenyl)prop-2-yn-1-ol
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
(1R,2S,4R)-N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
9-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
3-{5-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-{2-ethyl-4-[2-(3-hydroxypropyl)-1H-1,3-benzodiazol-1-yl]phenyl}acetamide
(3S,5R)-N3-(6-methylpyridin-3-yl)-N5-(oxan-4-yl)piperidine-3,5-dicarboxamide
N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methoxypropanamide
2-methoxy-6-{[3-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]methyl}phenol
(2R,3R,6R)-3-(4-fluorophenyl)-5-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(4-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methoxy}phenyl)ethan-1-one
1-[(4aR,8aS)-1-[2-(3-chlorophenyl)acetyl]-decahydro-1,6-naphthyridin-6-yl]-2-phenoxyethan-1-one
methyl (1R,3S,3aR,6aS)-3-(2-chloro-3-hydroxy-4-methoxyphenyl)-1-ethyl-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-(adamantan-1-yl)-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperazine
4-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-[2-(3-fluorophenyl)ethyl]-2-(4-{4-[methyl(pyridin-2-ylmethyl)amino]piperidin-1-yl}phenyl)acetamide
3-({4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}methyl)pyrrolidin-3-ol
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)(2-phenoxyethyl)amine
5-ethyl-4-(4-methanesulfonylphenyl)-6-methylthieno[2,3-d]pyrimidine
2-cyclopentyl-8-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
8-[(2-ethyl-1,3-thiazol-4-yl)methyl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl({[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})(thiophen-3-ylmethyl)amine
(5S,9aS,9bS)-5-(4-ethylphenyl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(2,3-dihydroxypropyl)-2-(4-fluorophenyl)-N-methylimidazo[1,2-a]pyridine-6-carboxamide
2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-(2,3-dihydro-1H-inden-2-yl)acetamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-1H-pyrazole-3-carboxamide
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-(6-chloropyridin-3-yl)-8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
3-[4-(benzenesulfonyl)phenyl]propanamide
(1-{2-[(3-chlorophenyl)methyl]-1,3-benzoxazole-6-carbonyl}piperidin-4-yl)methanol
1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-ethyl-8-methyl-2-(2-methylpyrimidin-5-yl)-N-(pyridin-4-ylmethyl)quinoline-4-carboxamide
7-{4-[(2-fluorophenyl)methyl]piperazine-1-carbonyl}-1,3-diazepane-2,4-dione
6,7-dimethoxy-3-({[1-(methoxymethyl)cyclopropyl](methyl)amino}methyl)-1,2-dihydroquinolin-2-one
4-{1-[(3-chlorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-5-methyl-1-(prop-2-en-1-yl)-1H-pyrazole
N-[2-(1H-imidazol-4-yl)ethyl]-6-(4-methoxyphenyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(cyclohexylmethyl)-N5-[(3,4-difluorophenyl)methyl]-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-(3-fluorophenyl)-N-{[8-(pyridin-4-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
2-[(2-ethyl-4-methyl-3-oxopiperazin-1-yl)methyl]-3,5-dimethoxybenzoic acid
2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenyl)-3,4,5,6,7,8-hexahydroquinazolin-4-one
4-(3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}phenyl)-4H-1,2,4-triazole
2-[2,4-dioxo-1-(2-phenylethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
3-(4-fluorophenyl)-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1H-pyrazole-5-carboxamide