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1-(2,3-dihydro-1H-inden-2-yl)-4-{imidazo[1,2-a]pyridine-3-carbonyl}-1,4-diazepane
N-(3-methoxypropyl)-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2,5-dimethoxyphenyl)methyl]acetamide
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-cyclopropyl-3-{[2-(dimethyl-1,3-thiazol-2-yl)ethyl]sulfamoyl}benzamide
4-methyl-6-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}-2-(pyridin-3-yl)pyrimidine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
1-{[3-(2-phenylethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}pyrrolidin-2-one
8-[(4-chloro-3-fluorophenyl)methyl]-2-(dimethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]propanamide
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N,1-dimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1H-imidazole-5-carboxamide
{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
1-[2-(4-methylpiperidin-1-yl)acetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-ethyl-5-[(4-hydroxypiperidin-1-yl)methyl]-N-(2-methylprop-2-en-1-yl)-1,2-oxazole-3-carboxamide
2-{2-[4-(hydroxymethyl)piperidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
N-(5-chloro-2-methoxyphenyl)-3-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-3-yl}propanamide
3-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-N-phenylpropanamide
4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]benzamide
7-hydroxy-2-oxo-4-[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]-1,2,3,4-tetrahydroquinoline-6-carboxylic acid
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-methylphenyl)methyl]piperidine
N-[1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2-phenylacetamide
(3S,4S)-1-[(4-cyanophenyl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
1-{1-[1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-4-yl]piperidin-3-yl}ethan-1-one
2-hydroxy-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-4-(methylsulfanyl)butanamide
3-(4-chloro-1H-pyrazol-1-yl)-1-(4-cyclohexyl-1,4-diazepan-1-yl)propan-1-one
{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
3-{[5-(1-cyclopentyl-1H-imidazol-2-yl)furan-2-yl]sulfanyl}-4-methyl-4H-1,2,4-triazole
N-methyl-N-{2-phenyl-1-[1-(quinolin-4-ylmethyl)piperidin-4-yl]ethyl}thiophene-2-carboxamide
N,2,7-trimethyl-N-(quinolin-5-ylmethyl)pyrazolo[1,5-a]pyrimidine-5-carboxamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-6-methylimidazo[1,2-a]pyridine-2-carboxamide
1-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]-4-(3-chlorophenyl)piperazine
3-{1-[4-(4-hydroxyphenyl)butan-2-yl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
6-[(3,5-dimethoxyphenyl)methoxy]-4-(2-methyl-1H-1,3-benzodiazole-6-carbonyl)-1-(propan-2-yl)-1,4-diazepan-2-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-3-(2-oxoazepan-1-yl)propanamide
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(2,4-dimethoxyphenyl)ethyl]amine
N-cyclopentyl-N-({3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-2-(trifluoromethyl)benzamide
1-[(3-methoxyphenyl)methyl]-5-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]piperidin-2-one
5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-methyl-N-(oxolan-3-yl)-1H-pyrazole-4-carboxamide
1-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}urea
2-[4-(6-methoxypyridin-3-yl)-3,5-dimethyl-1H-pyrazol-1-yl]-N-(1-methyl-1H-indazol-3-yl)acetamide
2-(4-methoxyphenoxymethyl)-4-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1,3-oxazole
methyl (2S,4R)-4-(2,3-dimethyl-1H-indole-7-amido)-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]pyrrolidine-2-carboxylate
2-methoxy-3-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridine
[7-(1-methyl-1H-imidazol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
3-[5-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-N-(propan-2-yl)propanamide
(1S,5R)-3-(pyridin-3-ylmethyl)-6-[(2,4,5-trimethylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}propan-1-one
(2S,4S)-4-amino-N-methyl-1-(4-phenoxybutanoyl)pyrrolidine-2-carboxamide