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4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-{[4-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
4-{[6-(2,5-dimethoxyphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}thiomorpholine
2-methyl-2-[2-(2-methyl-1,4-oxazepan-4-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]propanoic acid
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-1,4-diazepane
N-(3-{5-methyl-4-[(1,3-thiazol-4-ylformamido)methyl]-1,3-oxazol-2-yl}phenyl)pyridine-2-carboxamide
4-ethyl-3-{1-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(dimethyl-1,3-oxazol-4-yl)methyl]-6-[(dimethylamino)methyl]pyrimidin-4-amine
N-[3-(4-chlorophenoxy)-2-hydroxypropyl]-1-ethyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-{4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-cyclopentyl-3-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}piperidine
3-(3-chlorobenzoyl)-N-(2-methoxy-5-methylphenyl)piperidine-1-carboxamide
2,4-dimethyl-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)pyrimidine-5-carboxamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(4-methylpyrimidine-5-carbonyl)pyrrolidin-3-yl]methanol
N-[(2R,3R)-2-(benzyloxy)-1'-[(6-methylpyridin-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
5-[1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
4-{4-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
N-[3-(4-{[(4-methoxyphenyl)methyl]amino}piperidin-1-yl)phenyl]pyridine-3-carboxamide
2-{5-[(4-methylpiperazin-1-yl)methyl]pyridin-2-yl}benzonitrile
3-(3-hydroxy-3-methylbutyl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]benzamide
2-[4-(1H-1,3-benzodiazol-2-ylmethyl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
N-[2-(3-fluorophenyl)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
N-[(4-fluorophenyl)methyl]-N-(2-methoxyethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-(4-fluorophenyl)-4-[2-(propan-2-yl)pyrimidine-5-carbonyl]piperazin-2-one
5-{4-hydroxy-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
N-[3-({cyclopentyl[2-(dimethylamino)ethyl]carbamoyl}amino)phenyl]-N-methylacetamide
N-[(6-hydroxypyrimidin-4-yl)methyl]-2-(4-phenylpiperidin-1-yl)acetamide
9-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
dimethyl({1-[3-(pyrazin-2-yl)phenyl]ethyl})amine
[1-(5-fluoro-1H-indole-2-carbonyl)-4-[(3-methoxyphenyl)methyl]piperidin-4-yl]methanol
N,N-dimethyl-1-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}pyrrolidin-3-amine
N-{2-methyl-4-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]phenyl}furan-2-carboxamide
3-{[4-(3-chlorophenyl)-5-({methyl[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amino}methyl)-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
6-methoxy-2-oxo-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-[2-(2,4-difluorophenyl)-1-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
2-methyl-N-{3-[5-methyl-4-({2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamido}methyl)-1,3-oxazol-2-yl]phenyl}furan-3-carboxamide
(3aS,6aS)-1-[2-(benzyloxy)benzoyl]-octahydropyrrolo[2,3-c]pyrrole
1-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(1H-imidazol-1-yl)ethan-1-one
N-[3-(cyclohexylsulfanyl)propyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2-chloro-4-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
1-phenyl-5-{5-phenyl-1H-pyrazolo[3,4-b]pyridin-6-yl}-1H-pyrazole
8-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-methylacetamide
1-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]-4-methyl-1,4-diazepane
1-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-4-methylpiperidine-4-carbonitrile
2-(1,2-benzoxazol-3-yl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
N-(1-methyl-3-{1-[2-(morpholin-4-yl)propyl]-1,2,5,6-tetrahydropyridin-3-yl}-1H-pyrazol-5-yl)acetamide
8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-ethyl-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-(3-methylphenyl)ethan-1-one
2-(4-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol