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(2R)-1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}pyrrolidine-2-carboxamide
N-(2-{7-[(2,3-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2,4-dimethylbenzamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(E)-2-phenylethenesulfonamido]acetic acid
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-4-(propan-2-yloxy)benzamide
1-{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}piperidine-3-carboxamide
N-[2-(1-hydroxycyclopentyl)ethyl]-N-methyl-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
N-[1-(3-methylpyridin-2-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N,N-diethyl-1-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)pyrrolidin-3-amine
1-[1-(2-cyclopropylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-4-ol
{[4-ethoxy-3-(prop-2-en-1-yl)phenyl]methyl}(methyl)[1-(pyridin-3-yl)ethyl]amine
4-{[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]methyl}pyridine
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2-(5-methyl-1,2-oxazol-3-yl)piperidine
2-(4-phenylpiperidin-1-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
2-{2-[2-(4-ethylpiperazin-1-yl)ethoxy]phenyl}-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
(2S)-2-(dimethylamino)-1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-phenylpropan-1-one
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
[(3R,4S)-1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-[(1S,5R)-6-(3-ethyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-{5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl}propanamide
3-(2-methyl-1H-imidazol-1-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
(4-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)methanol
1-{4-[4-(4-fluorophenyl)-4-hydroxypiperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
4-(5-chlorothiophen-2-yl)-5-(propan-2-yl)pyrimidine
2-amino-4-(2,1,3-benzoxadiazol-4-yl)-6-(trimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-{2-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}ethan-1-one
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
N-[(2-fluorophenyl)methyl]-5-{[(4-methoxyphenyl)methyl]amino}-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-butyl-1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-3-carboxamide
5-{[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
(3S,4R)-4-methyl-1-[5-(propan-2-yl)pyrimidin-4-yl]piperidine-3,4-diol
1-ethyl-3,5-dimethyl-4-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]-1H-pyrazole
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]piperidine-3-carboxamide
3-[(2R,3R,6R)-5-(4-methoxybenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
3-(methylsulfanyl)-1-[3-(2-phenylethyl)piperidin-1-yl]propan-1-one
(3R,4R)-1-(4-fluoro-3-methylbenzoyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
5-butyl-4-(4-ethoxypiperidin-1-yl)-6-methylpyrimidin-2-amine
9-[(2R)-2-cyclohexyl-2-hydroxyacetyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-N-methylbutanamide
4-(4-methyl-1H-imidazole-2-carbonyl)-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
1-(2-{4-[(2-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-3-methoxy-1,2-dihydropyridin-2-one
N-(4-methoxy-2-methylphenyl)-2-[2-(morpholin-4-yl)ethyl]piperidine-1-carboxamide
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperidin-3-amine
methyl 5-[3-(1H-pyrazol-4-yl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-(2-hydroxyethyl)-4-[4-(3-methylphenoxy)piperidin-1-yl]pyridine-2-carboxamide
6-(3-chlorophenyl)-N-(2-methoxyethyl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-{5-[4-methoxy-3-(methoxymethyl)phenyl]-4-phenyl-1H-imidazol-1-yl}-N-methylacetamide
4-[(2,2-dimethylpiperazin-1-yl)methyl]-N-(2-propyl-2H-1,2,3-triazol-4-yl)benzamide
6-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
(3R,4R)-4-methyl-3-(propan-2-yl)-1-(2,2,3,3-tetramethylcyclopropanecarbonyl)pyrrolidin-3-ol
N-[2-(2-fluorophenyl)-1-[1-(quinoxalin-5-ylmethyl)piperidin-4-yl]ethyl]-N-methylthiophene-2-carboxamide