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N-[2-(azepan-1-yl)-2-phenylethyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-[4-(4-{4-ethyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2,5-dioxoimidazolidin-4-yl}piperidine-1-carbonyl)phenyl]acetamide
1-[(3,5-dimethylphenyl)methyl]-4-(1-propanoylpyrrolidine-2-carbonyl)piperazin-2-one
2-(3,4-dimethoxyphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
1-cyclopropyl-4-[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
3-(ethoxymethyl)-1-methyl-5-[4-(pyrrolidin-1-yl)phenyl]-1H-1,2,4-triazole
3-(propan-2-yl)-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2-oxazole-5-carboxamide
1-methanesulfonyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
2-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-6-methylpyridine-3-carbonitrile
(3aR,6aR)-2-cyclopentyl-5-(2-ethoxy-2-oxoethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[1-(1-benzylpiperidin-4-yl)-2-(2,4-difluorophenyl)ethyl]-N-methylfuran-2-carboxamide
5-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-2-fluorobenzamide
1-(4-fluorophenyl)-4-{1-[1-(propan-2-yl)piperidine-4-carbonyl]piperidin-3-yl}piperazine
2-benzyl-3-methyl-4-[2-(methylsulfanyl)phenyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[3-(2-chlorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(quinoxalin-6-ylmethyl)acetamide
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](methyl)[1-(pyrimidin-4-yl)ethyl]amine
N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-1H-pyrazole-4-carboxamide
N-cyclohexyl-2-ethyl-N-[2-(1H-indol-3-yl)ethyl]pyrimidine-5-carboxamide
6-{[5-(morpholin-4-ylmethyl)quinolin-8-yl]oxy}pyridine-2-carbonitrile
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-(piperidin-1-yl)pyridine-3-carboxamide
8-benzyl-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4R)-1-{5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-methylpiperidine-3,4-diol
14-(2-methoxypyridin-3-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(pyridin-3-yl)piperazin-1-yl]butan-1-one
3-amino-1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-4-[4-(trifluoromethyl)benzenesulfonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(4-{[3-(5-methylfuran-2-yl)phenyl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
ethyl 1-[(2,5-dimethoxyphenyl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
2-(3-methoxyphenyl)-1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}piperidine
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}pent-4-en-1-one
2-(diethylamino)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}acetamide
9-(cyclopropylmethyl)-4-[3-(1H-imidazol-1-yl)propyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-4-(thiophen-2-yl)butanamide
(4S)-1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-(methoxymethyl)piperidine
2-cyclopropyl-N-[(1R)-1-(4-fluorophenyl)ethyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-{[7-chloro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(furan-2-ylmethyl)propanamide
1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
N-(2-methoxyethyl)-5-{1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-[2-(4-ethylmorpholin-2-yl)ethyl]-2-(1-methyl-1H-indol-3-yl)acetamide
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}ethan-1-one
N-(oxolan-2-ylmethyl)-3-(5-phenyl-1,3,4-oxadiazol-2-yl)-N-propylpropanamide
2-[1-(3-methylbutyl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl]ethan-1-ol
4-{[1-(ethylcarbamoyl)piperidin-4-yl]amino}pyrimidine-5-carboxylic acid
4-(3,6-dimethylpyrazin-2-yl)-2-{[4-(2-methylphenyl)piperazin-1-yl]methyl}phenol
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide