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N-ethyl-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}pyridine-4-carboxamide
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}naphthalene-1-sulfonamide
2-[2-(3-fluorophenyl)piperidine-1-carbonyl]benzonitrile
N,N-dimethyl-2-[2-(2-methylpropoxy)phenyl]pyridine-3-carboxamide
(4aR,7aS)-1-ethyl-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2,6-dimethylquinoline-4-carboxamide
N-{[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]methyl}-1H-indole-2-carboxamide
3-(2-methyl-1H-imidazol-1-yl)-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridazine
(2S,4R)-4-amino-N-methyl-1-{[1-(prop-2-en-1-yl)-1H-1,3-benzodiazol-2-yl]methyl}pyrrolidine-2-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
N-{2-[(E)-2-phenylethenyl]pyridin-3-yl}cyclopropanecarboxamide
N-{3-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidine-1-carbonyl]phenyl}acetamide
(2S)-3-(4-hydroxyphenyl)-2-{[1-(9H-purin-6-yl)piperidin-4-yl]amino}propanamide
(2E)-3-(2-chlorophenyl)-1-[4-(3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}phenoxy)piperidin-1-yl]prop-2-en-1-one
(5S,9aS,9bS)-2-methyl-5-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
methyl 2-{5-methyl-2-[(2-methylbutanamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}benzoate
(3aR,6aR)-N-(cyclohex-1-en-1-ylmethyl)-2-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(1S,5R)-6-benzyl-3-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
[1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3-propylpiperidin-3-yl]methanol
N-[(3R,4R)-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
N-[(5-{[2-(3-methoxypropyl)piperidin-1-yl]methyl}furan-2-yl)methyl]-N-methylmethanesulfonamide
9-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(oxan-4-yl)-5-[(1R,2R)-2-phenylcyclopropyl]-1H-1,2,4-triazole
N-[3-(diethylamino)propyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(6-methylpyridin-2-yl)piperazine
5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-(2-methoxyethyl)-4-oxo-N-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3-carboxamide
3-methyl-4-[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(3aS,6aR)-3-[2-(pyridin-2-yl)ethyl]-5-(4,4,4-trifluorobutyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(methoxymethyl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}cyclobutane-1-carboxamide
3-(5-benzyl-1,3,4-thiadiazol-2-yl)-1-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
2-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)acetic acid
5,8-dimethyl-2-{[4-(pyrrolidin-3-yl)piperazin-1-yl]methyl}quinolin-4-ol
N-cyclopropyl-1-{1-[(3-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
9-[(2,5-dimethylphenyl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-6-oxo-1,6-dihydropyrimidine-5-carboxamide
3-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-imidazol-2-yl]-1,2-dihydroquinolin-2-one
3-[(3R,4S)-4-(dimethylamino)-1-(quinoline-4-carbonyl)piperidin-3-yl]propanoic acid
N-[(3R,4S)-1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
ethyl 2-{[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]amino}benzoate
1-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-phenyl-1H-pyrazole-5-carboxamide
4-fluoro-N-[(1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)methyl]benzamide
1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl][(2-fluoro-5-methoxyphenyl)methyl]methylamine
methyl 3-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-benzyl-N-[2-(dimethylamino)ethyl]-4-(piperidin-3-yl)benzamide
9-(5-fluoro-2-methoxybenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 6-[(3-chlorophenyl)methyl]-2-(ethylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
9-(4-chloro-3-fluorobenzoyl)-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
4-[(4-chloro-3-fluorophenyl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one