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4-(1-methyl-1H-imidazol-2-yl)-1-(oxolane-3-carbonyl)piperidine
1-[5-(oxolan-2-yl)thiophene-2-carbonyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2-methyl-6-(piperidin-3-yl)pyrimidin-4-amine
(3S,4R)-1-(3-chloropyridine-4-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
N-{[7-chloro-5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(thiophen-2-yl)butanamide
1-(cyclopropylmethyl)-5-(3-fluoro-4-methoxybenzoyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(cyclopropylmethyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-methyl-N-(pyridin-3-ylmethyl)-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoline
3-(2-methyl-1H-imidazol-1-yl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
N-({3,5-dimethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-2-(dimethyl-1,2-oxazol-4-yl)-N-(pyridin-4-ylmethyl)acetamide
methyl 3-[(1-methyl-1H-pyrazol-4-yl)methyl]-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
ethyl 1-methyl-5-({4-[methyl(phenyl)amino]phenyl}methyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-amino-1-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
2-[3-({4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)-2-methyl-1H-indol-1-yl]acetamide
1-[(2,2-dimethyloxan-4-yl)methyl]-4-(4-methoxybenzoyl)piperazine
5-(3,4-difluorophenoxymethyl)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
1-({3-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}methyl)azepane
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}propanamide
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
N-(2-{7-[(4-methoxy-2,3-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
N-cyclopropyl-3-(1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)propanamide
({4-ethyl-5-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
5-cyclopropanecarbonyl-1'-(3-ethyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(2-benzylmorpholine-4-carbonyl)-3,4,7-trimethyl-1H-indole
3-[(3S,4S)-1-ethyl-4-methoxypyrrolidin-3-yl]-1-[2-(4-fluorophenoxy)pyridin-3-yl]urea
2-(dimethyl-1,2-oxazol-4-yl)-1-(4-{5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)ethan-1-one
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
7-amino-4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
N-[(3-methoxyphenyl)methyl]-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(5-pentyl-1,3,4-thiadiazol-2-yl)-4-(pyridin-4-ylmethyl)piperazine-1-carboxamide
N-{[2-(3-chlorophenyl)-8-methylquinolin-3-yl]methyl}-N-cyclopropylacetamide
2-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoline
3-(1-methyl-1H-imidazole-2-carbonyl)-1-(thiophen-3-ylmethyl)piperidine
9-methoxy-3-[(3-methoxyphenyl)methyl]-N-methyl-7-oxo-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-[1-(methylcarbamoyl)cyclohexyl]benzamide
1-{3-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}ethan-1-one
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
4-[1-(1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]morpholine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(4-phenylpiperidin-1-yl)acetamide
2-{[3-(2-ethylphenoxy)azetidin-1-yl]methyl}benzoic acid
1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
[1-(1-cyclopentanecarbonylpiperidin-3-yl)piperidin-4-yl]methanol
N-[(3R,4S)-4-cyclopropyl-1-(3-fluoropyridin-4-yl)pyrrolidin-3-yl]-2-methoxy-2-methylpropanamide
3-[(cyclopentylmethyl)(methyl)amino]-N-methylbutanamide
6-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-N,N-dimethylpyrazine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
4-[2-methoxy-5-(propan-2-yl)phenyl]-1-[(2S)-oxolan-2-ylmethyl]-1H-1,2,3-triazole
1-[3-(cyclohexylsulfanyl)propyl]-3-[3-(2-oxopyrrolidin-1-yl)phenyl]urea
4-(1-ethyl-1H-imidazol-2-yl)-N-(3-ethylphenyl)piperidine-1-carboxamide