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1-(4-chloro-1H-pyrazole-3-carbonyl)-4-(2-methoxybenzoyl)piperazine
1-[(2,6-difluorophenyl)methyl]-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-(methylamino)-2-phenylethan-1-one
4-({4-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)piperazine-1-carboxamide
8-fluoro-4-oxo-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,4-dihydroquinoline-3-carboxamide
1-[2-amino-6-(dimethylamino)pyrimidin-4-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(3aR,5S,6S,7aS)-2-(1,3,4-thiadiazol-2-yl)-octahydro-1H-isoindole-5,6-diol
3-(4-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}benzenesulfonyl)propanoic acid
N'-cyclopentyl-N-methyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]butanediamide
({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
2-(diethylamino)-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethan-1-one
4-[2-(cyclopropylmethyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1-(propan-2-yl)pyrrolidin-2-one
ethyl 4-{[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]amino}piperidine-1-carboxylate
N'-[(4-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethoxy}-3-methoxyphenyl)methyl]-N,N-dimethyl-N'-[(3S)-2-oxoazepan-3-yl]butanediamide
2-(2-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-{4-[3-(4-chloro-2-methylbenzoyl)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}oxolane-3-carboxamide
8-chloro-2-({[2-(dimethylamino)ethyl](oxolan-2-ylmethyl)amino}methyl)quinolin-4-ol
4-(morpholin-4-yl)-6-(pyrimidin-5-yl)pyrimidin-2-amine
9-methoxy-7-(6-methoxypyridazin-3-yl)-4-[4-(1H-pyrazol-1-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2E)-1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-(1H-imidazol-4-yl)prop-2-en-1-one
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl)[(5-methylfuran-2-yl)methyl]amine
(4aR,8aS)-6-{[4-(2-methylphenyl)phenyl]methyl}-1-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
4-{[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazin-1-yl]methyl}-2-methoxyphenol
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-1-methyl-1H-indole-2-carboxamide
2-cyclopentyl-1-[3-(3-{[methyl(1-methylpiperidin-4-yl)amino]methyl}phenoxymethyl)piperidin-1-yl]ethan-1-one
N-[4-methyl-2-(3,4,5-trimethoxyphenyl)phenyl]propanamide
5-methoxy-2-[3-(3-methoxyphenoxy)azetidin-1-yl]pyrimidine
1-(4-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
4-(2-methyl-1H-imidazol-1-yl)-1-(2-methylfuran-3-carbonyl)piperidine-4-carboxylic acid
N-butyl-3-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-methyloxolane-2-carboxamide
N-[2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide
2-hydroxy-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
[9-(1H-imidazol-2-ylmethyl)-3-(pyrazin-2-yl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
N-{1-[4-(isoquinolin-5-yl)phenyl]ethyl}acetamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-methyl-N-(pyrimidin-4-ylmethyl)acetamide
3-methyl-4-[3-(propan-2-yl)-5-[(pyridin-3-yloxy)methyl]-1H-1,2,4-triazol-1-yl]pyridine
7-[(2,3-dimethoxyphenyl)methyl]-6-oxo-N-propyl-2,7-diazaspiro[4.5]decane-2-carboxamide
1-[3-chloro-4-(1H-imidazol-1-yl)phenyl]-3-[3-(pyrrolidin-1-yl)propyl]urea
2-(dimethylamino)-2-(4-fluorophenyl)-N-[(5-methoxy-1H-indol-2-yl)methyl]acetamide
5-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-N-propylpyrimidin-2-amine
3-{1-[2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]piperidin-3-yl}benzoic acid
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[3-(3-methylphenoxymethyl)piperidin-1-yl]propan-1-one
3-(2-amino-1,3-thiazol-4-yl)-1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}propan-1-one
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
1-{1-[2-(methylamino)pyridine-4-carbonyl]piperidin-4-yl}-2-phenylethan-1-ol
3-[2-(dimethylamino)ethyl]-5-[1-(4-methylbenzoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
N'-(2-ethoxyphenyl)-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]propanediamide
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine