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1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
4-{1-[3-(3-fluorophenyl)phenyl]piperidin-4-yl}-1,4-oxazepane
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1-phenylcyclohexane-1-carboxamide
2-acetyl-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylbenzamide
[(5-ethylfuran-2-yl)methyl](methyl)[2-(pyridin-4-yl)ethyl]amine
N-cyclohexyl-2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]butanamide
(3S,4R)-4-(3-fluorophenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxylic acid
2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
N-methyl-2-(5-methyl-3-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonane-7-carbonyl}-1H-pyrazol-1-yl)acetamide
N-[2-(2,4-difluorophenyl)-1-(1-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}piperidin-4-yl)ethyl]-N-methylpropanamide
(1S)-1-[3-methyl-1-(naphthalen-1-yl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
6-[3-(2-hydroxyethyl)-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl]pyridine-2-carbonitrile
N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2,2,3,3-tetramethylcyclopropane-1-carboxamide
3-{2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
(4aR,8aS)-1-[3-(dimethylamino)propyl]-6-(pyridin-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(5-fluoro-2-methylphenyl)methyl]benzamide
N-methyl-1-[(2E)-3-phenylprop-2-en-1-yl]-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
[(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl){[6-(trifluoromethyl)pyridin-3-yl]methyl}amine
N-methyl-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
6-(2,5-dimethylfuran-3-yl)-7-(prop-2-en-1-yl)-2-(pyrrolidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
4,6-dimethyl-2-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)pyridine-3-carbonitrile
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{4-[2-(3-methoxyphenyl)-1-[methyl(pyridin-2-ylmethyl)amino]ethyl]piperidin-1-yl}propan-1-one
1-benzyl-N-ethyl-4-oxo-5-(4-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
methyl (2S)-3-methyl-2-{3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamido}butanoate
N-benzyl-N-[(3-methylpyridin-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N-({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-3-yl}methyl)-2-hydroxypyridine-3-carboxamide
{7-[3-(4H-1,2,4-triazol-4-yl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
1-[(3-methylpyridin-2-yl)methyl]-4-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperazine
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-acetamidobenzamide
2-(4-{[3-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}phenoxy)acetic acid
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(propan-2-yl)amino]methyl}piperidin-2-one
N-ethyl-1,3-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-5-(pyridine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[1-(2,2-diphenylethyl)piperidin-3-yl]-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
3-hydroxy-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
(3S)-1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-N,N-dimethylazepan-3-amine
3-[1-(2-amino-6-hydroxypyrimidin-4-yl)piperidin-4-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methoxy-N-[2-(1,2,5-thiadiazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
8-(2,4-dimethoxypyrimidin-5-yl)quinoline
5-[(dimethylamino)methyl]-N-[3-(furan-2-yl)propyl]furan-2-carboxamide
(5S)-5-(3,3-diphenylpiperidine-1-carbonyl)pyrrolidin-2-one
5-({1-[4-(furan-2-yl)phenyl]piperidin-4-yl}amino)-1-methylpiperidin-2-one
2-(2-fluorophenyl)-5-(1H-pyrazol-1-ylmethyl)-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
2-(3-methoxypropyl)-9-(quinolin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{1-[(3-fluorophenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
1,6-dimethyl-3-[2-methyl-4-(2-methylpropyl)-3-oxopiperazine-1-carbonyl]-1,4-dihydroquinolin-4-one
(3S,4R)-4-phenyl-1-[(2,3,4-trimethoxyphenyl)methyl]pyrrolidine-3-carboxylic acid