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2-{2-[1-(2-methoxyethyl)piperidin-4-yl]-1H-imidazol-1-yl}propan-1-ol
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-6-methylpyridine-3-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(1H-indol-4-ylmethyl)-5-methoxybenzamide
N-[(4-hydroxyphenyl)methyl]-2-(3-phenylpiperidin-1-yl)acetamide
3-{[1-(3-methylphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
4'-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(1R,3S)-7-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-7-azaspiro[3.5]nonane-1,3-diol
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
1-[(2-chlorophenyl)methyl]-N-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-[(3-fluorophenyl)methyl]-4-[5-(oxolan-2-yl)thiophene-2-carbonyl]piperazine
3-fluoro-N-{[7-(2,5,7-trimethylquinoline-4-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
4-(cyclopropylmethyl)-1-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,4-diazepan-5-one
(R)-cyclohexyl({1-[2-(1H-imidazol-5-yl)ethyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl})methanol
1-{[(3R,4R)-1-[(2,4-dimethoxy-3-methylphenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
2-(5-{[2-(aminomethyl)morpholin-4-yl]methyl}furan-2-yl)benzonitrile
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(2-cyclohexylpyrimidin-5-yl)methyl]pyrrolidin-3-yl]methanol
N-[2-({5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazol-4-yl}formamido)ethyl]acetamide
5-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
5-[(2-chlorophenyl)methyl]-5-[1-(3,5-dimethylbenzoyl)piperidin-4-yl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
7-[(3-methylphenyl)methyl]-2-(1-methylpiperidine-4-carbonyl)-2,7-diazaspiro[4.5]decane
1-[2-(4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-1,2,3-triazol-1-yl)ethyl]piperidine
N-cyclopropyl-N-{[3-(oxolan-2-ylmethoxy)phenyl]methyl}-2-(trifluoromethyl)benzamide
2,6-dimethyl-5-{2-oxo-2-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-3,4-dihydropyrimidin-4-one
N-(1-{1-[2-(2,5-difluorophenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
1-benzyl-2-methyl-3-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]-4,5,6,7-tetrahydro-1H-indol-4-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-2-one
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-5-methanesulfonyl-2-methylpyrimidin-4-amine
2-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
2-(5-{[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
7-(cyclohex-3-en-1-ylmethyl)-4-(morpholin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[(thiolan-3-yl)amino]pyridine-3-carboxamide
2-[4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]benzonitrile
(1S,4S)-N,3,3-trimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-methylidenebicyclo[2.2.1]heptane-1-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}propanamide
4-[3-(2-methoxyphenoxy)azetidin-1-yl]pyrimidine-5-carboxylic acid
8-(3-hydroxybenzoyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(3-fluorophenyl)-N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
6-(4-hydroxybutan-2-yl)-1-[(4-methoxyphenyl)methyl]-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-methoxy-4-[(1E)-3-{4-[5-(propan-2-yl)pyrimidin-4-yl]piperazin-1-yl}prop-1-en-1-yl]phenol
1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidine
7-[(4-fluorophenyl)methyl]-2-(1,3-thiazol-2-yl)-2,7-diazaspiro[4.5]decane
1-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methylhexanamide
3-[(oxan-4-yl)sulfamoyl]-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
1-ethyl-4-{1-[3-(4-fluorophenyl)phenyl]piperidin-4-yl}piperazine
N-[4-(2-fluorophenoxy)phenyl]-1-(oxan-4-yl)piperidine-4-carboxamide
N,N-dimethyl-1-(2-methylpropyl)-5-{[2-(propan-2-yloxy)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(hydroxymethyl)-1-(5-methyl-4-phenylthiophene-3-carbonyl)piperidin-3-ol
N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide