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N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2-[2,6,6-trimethyl-4-oxo-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
1-(2-methoxyethyl)-3-(2-phenylethyl)-8-{[2-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-methoxy-N,3-dimethyl-N-[1-(pyridin-3-yl)pentyl]-1-benzofuran-2-carboxamide
{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[2-(furan-2-yl)pyrimidin-5-yl]methyl})methylamine
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-N-(3-methylphenyl)acetamide
N-[(3-methoxyphenyl)methyl]-4-methyl-N-(prop-2-en-1-yl)pyridine-3-carboxamide
7-methyl-2-{2-[3-(trifluoromethyl)phenyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
N-(2-chloro-6-methylphenyl)-3-(6-methoxynaphthalene-2-carbonyl)piperidine-1-carboxamide
9-(1-ethyl-1H-pyrazole-5-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
6-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]pyrazine-2-carboxamide
2-[1-(2,4-dimethylpyrimidine-5-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
4-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]benzene-1-sulfonamide
N-[1-(hydroxymethyl)cyclopentyl]-4-pentanamidobenzamide
7-methyl-3-{[1-(2-methylphenyl)-1H-pyrrol-2-yl]methyl}-3,7,11-triazaspiro[5.6]dodecan-12-one
4-(2,3,4-trimethoxyphenyl)thiophene-2-carboxamide
2-(2-methyl-1H-1,3-benzodiazol-5-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
2-(2-chloro-4-fluorophenoxymethyl)-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
2-(3,4-difluorophenyl)-5-(1H-imidazol-2-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-methylpyridazine
3-{1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(3-methyloxetan-3-yl)methyl]acetamide
N,N-dimethyl-2-(4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)acetamide
3-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-N-methylpyridin-2-amine
N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-4-(2-oxopyrrolidin-1-yl)benzamide
N-(1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperidin-4-yl)acetamide
5-amino-3-[4-(1H-pyrazol-1-yl)phenyl]-1,6-diazatricyclo[6.2.2.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
5-(methoxymethyl)-N-({3-methyl-7-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
3-(2-hydroxyphenyl)-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
8-{[3-(5-methylfuran-2-yl)phenyl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
3-({2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)phenol
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
1-[(4-methylphenyl)methyl]-4-[2-(propylsulfanyl)acetyl]piperazin-2-one
1-{2-[(1-benzylpiperidin-4-yl)amino]ethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrrolidine-2-carboxamide
(3R)-1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-ol
N-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
(4aS,8aR)-1-butyl-6-(pyridazine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
5-tert-butyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-1,3,4-oxadiazol-2-amine
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)propanamide
methyl[(2-methyl-1,3-thiazol-4-yl)methyl]{[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}amine
(1R,5R)-6-(cyclobutylmethyl)-3-(3-ethyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-benzyl-1-[(3-methylpyridin-2-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)-2,3-dihydro-1-benzofuran-2-carboxamide
methyl 4-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-4-oxobutanoate
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
ethyl 4-(2-methoxyethyl)-1-{1-[3-(trifluoromethyl)phenyl]propan-2-yl}piperidine-4-carboxylate
5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-1-methyl-1,2-dihydropyridin-2-one
N-[4-({3-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}methyl)phenyl]acetamide
N-methyl-1-(7-methyl-1-benzofuran-2-carbonyl)-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine