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5-[(2,3-dichloro-6-fluorophenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-benzyl-8-[(6-methylpyridin-2-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,5R)-1-(3-methoxypropanoyl)-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
2-methyl-5-(3-methylphenyl)-4-{1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}pyrimidine
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[2-(1H-pyrazol-1-yl)acetyl]-1,4-diazepan-5-one
2-(dimethylamino)-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-2-(3-methylphenyl)acetamide
1-(4-benzylpiperidin-1-yl)-3-[1-(oxolane-2-carbonyl)piperidin-4-yl]propan-1-one
ethyl 5-[(2S)-5-oxopyrrolidine-2-carbonyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-hydroxy-N-[(2-methoxyphenyl)methyl]-2-methyl-N-[(2-methylphenyl)methyl]pyrimidine-5-carboxamide
2-ethyl-4-phenyl-9-(1H-pyrrole-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
3-(1,3-thiazol-2-yl)quinoline
1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]ethan-1-one
N-{[2-(benzyloxy)phenyl]methyl}-1-ethylpyrrolidine-3-carboxamide
2-{[2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-4,6-dimethylpyrimidine
N-methyl-2-(1-propylpiperidin-4-yl)-N-[1-(1,3-thiazol-5-yl)ethyl]acetamide
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-[methyl(piperidin-4-yl)amino]ethan-1-one
1-(4-{[(oxan-4-yl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
4-[(2-methylphenyl)sulfanyl]-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
5-[2-(4-chlorophenyl)morpholine-4-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
(1-methyl-5-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
2-methyl-1-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-6-(methoxymethyl)pyridine
N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
N,2,7-trimethyl-N-[1-(pyridin-2-yl)ethyl]quinoline-4-carboxamide
3-[1-(1-acetylpiperidin-4-yl)-1H-pyrazol-5-yl]-1-(3-fluorophenyl)urea
N-cyclopropyl-5-methyl-4-{[1-(thiophen-2-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
6-(1-benzofuran-2-ylmethyl)-N-[4-(methylsulfanyl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
3-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-5-(3-fluorophenyl)-1,2,4-triazine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-5-propyl-1,2-oxazole-3-carboxamide
1-(4-{[2-(dimethylamino)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-3-(1H-pyrazol-1-yl)propan-1-one
1-(4-fluorophenyl)-5-[(2-methoxyethoxy)methyl]-3-methyl-1H-1,2,4-triazole
6-amino-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]pyridine-3-carboxamide
N-ethyl-5-[2-(4-methylpentyl)morpholine-4-carbonyl]pyrimidin-2-amine
2-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2,9-diazaspiro[5.5]undecan-3-one
(3R,5S)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(piperidin-1-yl)piperidine
2-methyl-N-({8-[(2,4,5-trimethylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)propanamide
8-methoxy-2-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}quinoline
4-[(2-fluoro-4,5-dimethoxyphenyl)methyl]piperazine-2-carboxylic acid
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(5-oxopyrrolidin-2-yl)acetamide
7-(5-chloropyridin-2-yl)-4-(pyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-4-carboxamide
3-ethyl-4-[4-(4-hydroxybut-1-yn-1-yl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
6-[(diethylamino)methyl]-N-(oxolan-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N,1,3-trimethyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
6-fluoro-2-({4-[2-(morpholin-4-yl)ethyl]piperazin-1-yl}methyl)quinolin-4-ol
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
4-(2-methyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
ethyl 1-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}-4-(3-phenylpropyl)piperidine-4-carboxylate